SCHEMBL22719910

SCHEMBL22719910

CC1(C)OCc2c(COc3ccc(F)cc3)cnc(C#N)c2O1

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.41
KMT2A Q03164 2/20 0.41
MAPK1 P28482 2/20 0.41
TSHR P16473 6/20 0.39
L3MBTL1 Q9Y468 3/20 0.39
MAPT P10636 6/20 0.37
NPSR1 Q6W5P4 2/20 0.37
HTT P42858 2/20 0.37
MEN1 O00255 1/20 0.37
GAA P10253 4/20 0.35
MAOB P27338 1/20 0.33
KDM4E B2RXH2 1/20 0.33
LMNA P02545 2/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
TP53 P04637 2/20 0.32
HPGD P15428 2/20 0.32
GRM5 P41594 1/20 0.32
ALOX15 P16050 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22283910 0.84 ALDH1A1 (0.59) ALDH1A1KMT2AMAPK1MAPTGAA
SCHEMBL22719897 0.81 ALDH1A1 (0.41) ALDH1A1KMT2AMAPK1L3MBTL1MEN1
SCHEMBL22719962 0.81 KMT2A (0.41) ALDH1A1KMT2AMAPK1MAPTMEN1
SCHEMBL3442472 0.81 KMT2A (0.57) ALDH1A1KMT2AMAPK1MAPTMAOB
SCHEMBL30193078 0.79 KMT2A (0.40) ALDH1A1KMT2AMAPK1L3MBTL1MAPT
SCHEMBL1503189 0.79 KMT2A (0.40) ALDH1A1KMT2AMAPK1L3MBTL1MAPT
SCHEMBL22719912 0.78 KMT2A (0.39) ALDH1A1KMT2AMAPK1TSHRMAPT
SCHEMBL22719947 0.75 LMNA (0.46) ALDH1A1KMT2AMAPK1TSHRGAA
SCHEMBL22719950 0.69 MAOB (0.39) ALDH1A1KMT2AMAPK1MAPTMAOB
SCHEMBL1503147 0.67 ALDH1A1 (0.39) ALDH1A1KMT2AMAPK1MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020237374-A1 PICOLINIC ACID DERIVATIVES AND USE THEREOF FOR TREATING DISEASES ASSOCIATED WITH ELEVATED CHOLESTEROL MONTREAL HEART INSTITUTE (CA) 2020-12-03 WO disclosed
WO-2020237374-A1 PICOLINIC ACID DERIVATIVES AND USE THEREOF FOR TREATING DISEASES ASSOCIATED WITH ELEVATED CHOLESTEROL MONTREAL HEART INSTITUTE (CA) 2020-12-03 WO disclosed