SCHEMBL22738232

SCHEMBL22738232

COC(=O)c1ncc(Cn2ccc3cc(I)ccc32)c2c1OC(C)(C)OC2

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.35
MAPK1 P28482 1/20 0.35
KMT2A Q03164 1/20 0.35
KRAS P01116 1/20 0.33
HCRTR1 O43613 1/20 0.33
HCRTR2 O43614 1/20 0.33
EPHX2 P34913 1/20 0.33
MAOB P27338 2/20 0.33
HDAC8 Q9BY41 3/20 0.32
HDAC6 Q9UBN7 3/20 0.32
HDAC11 Q96DB2 2/20 0.32
HDAC3 O15379 2/20 0.32
HDAC4 P56524 1/20 0.32
HDAC7 Q8WUI4 1/20 0.32
HDAC9 Q9UKV0 1/20 0.32
HDAC5 Q9UQL6 1/20 0.32
SYK P43405 1/20 0.32
MTNR1A P48039 2/20 0.32
MTNR1B P49286 2/20 0.32
AR P10275 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22738287 0.91 MTNR1A (0.41) ALDH1A1MAPK1KMT2AHCRTR1HCRTR2
SCHEMBL22738235 0.91 ALDH1A1 (0.37) ALDH1A1MAPK1KMT2AHCRTR1HCRTR2
SCHEMBL22719960 0.90 PPARG (0.38) ALDH1A1MAPK1KMT2AMAOB
SCHEMBL22719901 0.90 EGLN1 (0.35) ALDH1A1MAPK1KMT2AKRASHCRTR1
SCHEMBL22719944 0.85 HDAC1 (0.36) ALDH1A1MAPK1KMT2AHCRTR1HCRTR2
SCHEMBL22738309 0.83 EGLN1 (0.44) HCRTR1HCRTR2EPHX2HDAC8HDAC6
SCHEMBL22738238 0.82 ALDH1A1 (0.37) ALDH1A1MAPK1KMT2AHCRTR1HCRTR2
SCHEMBL22719930 0.81 PPARG (0.39) MAOB
SCHEMBL22719923 0.80 MTNR1A (0.40) ALDH1A1HDAC8HDAC6HDAC11HDAC3
SCHEMBL22719921 0.78 NPY5R (0.39) MAOB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020237374-A1 PICOLINIC ACID DERIVATIVES AND USE THEREOF FOR TREATING DISEASES ASSOCIATED WITH ELEVATED CHOLESTEROL MONTREAL HEART INSTITUTE (CA) 2020-12-03 WO disclosed