SCHEMBL2275016

SCHEMBL2275016

O=C(Nc1cc(-c2ccccc2)ccc1C(=O)O)c1cc(-c2ccccc2)n[nH]1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.58
CHEK1 O14757 1/20 0.57
RET P07949 1/20 0.57
PDGFRB P09619 1/20 0.57
PIM1 P11309 1/20 0.57
PDGFRA P16234 1/20 0.57
GSK3B P49841 1/20 0.57
RPS6KA3 P51812 1/20 0.57
LIMK1 P53667 1/20 0.57
CDK5 Q00535 1/20 0.57
TYRO3 Q06418 1/20 0.57
MAPK14 Q16539 1/20 0.57
LRRK2 Q5S007 1/20 0.57
AURKB Q96GD4 1/20 0.57
CLK4 Q9HAZ1 1/20 0.57
DYRK1B Q9Y463 1/20 0.57
ACLY P53396 1/20 0.56
MAPK8 P45983 3/20 0.55
ADORA3 P0DMS8 1/20 0.53
ADORA2A P29274 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2274064 0.84 TP53 (0.52) TP53CHEK1RETPDGFRBPIM1
SCHEMBL2271944 0.84 MAPT (0.55) TP53CHEK1RETPDGFRBPIM1
SCHEMBL2275453 0.81 ACLY (0.76) ACLYDHODHHDAC3HDAC1HDAC2
SCHEMBL2270222 0.81 DHODH (0.77) ACLYDHODHHDAC3HDAC1HDAC2
SCHEMBL6814323 0.80 SNCA (0.59) TP53CHEK1RETPDGFRBPIM1
SCHEMBL27716724 0.78 ACR (0.70) TP53CHEK1RETPDGFRBPIM1
SCHEMBL3844821 0.77 HDAC1 (0.67) TP53CHEK1RETPDGFRBPIM1
SCHEMBL1318089 0.77 ACLY (0.60) TP53ACLYDHODHHDAC1ALDH1A1
SCHEMBL2272508 0.77 ACLY (0.63) ACLYDHODHHDAC1ALDH1A1MAPT
SCHEMBL2270217 0.76 ACLY (0.58) ACLYDHODHHDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7999132-B2 Anthranilic acid derivative or salt thereof TOYAMA CHEMICAL CO., LTD. (JP) 2011-08-16 US disclosed
US-20090240052-A1 NOVEL ANTHRANILIC ACID DERIVATIVE OR SALT THEREOF TOYAMA CHEMICAL CO., LTD. (JP) 2009-09-24 US disclosed
EP-1820795-A1 NOVEL ANTHRANILIC ACID DERIVATIVE OR SALT THEREOF TOYAMA CHEMICAL CO., LTD. (JP) 2007-08-22 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090240052-A1 NOVEL ANTHRANILIC ACID DERIVATIVE OR SALT THEREOF MMP13, MMP26, MMP11 TP53 858/4885CHEK1 4352/4885RET 3447/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.