SCHEMBL2270217

SCHEMBL2270217

O=C(Nc1cc(-c2ccccc2)ccc1C(=O)O)c1cc(-c2ccccc2)ncn1

nearest known ligand 0.58

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ACLY P53396 8/20 0.58
KMO O15229 6/20 0.57
HDAC1 Q13547 1/20 0.50
SMO Q99835 1/20 0.50
MEN1 O00255 1/20 0.47
GFER P55789 1/20 0.47
KMT2A Q03164 1/20 0.47
SUCNR1 Q9BXA5 1/20 0.47
DHODH Q02127 1/20 0.47
GRIK1 P39086 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2275310 0.85 KMO (0.51) ACLYKMOSMOMEN1GFER
SCHEMBL2278060 0.85 KMO (0.51) KMODHODH
SCHEMBL1316823 0.84 ACLY (0.64) ACLYHDAC1SMOSUCNR1DHODH
SCHEMBL1317052 0.82 ACLY (0.64) ACLYHDAC1MEN1KMT2ASUCNR1
SCHEMBL1318089 0.81 ACLY (0.60) ACLYHDAC1SMOMEN1GFER
SCHEMBL13205947 0.80 ACLY (0.65) ACLYHDAC1SUCNR1GRIK1
SCHEMBL1316866 0.80 ACLY (0.62) ACLYHDAC1SMOMEN1KMT2A
SCHEMBL27716719 0.78 KMO (0.75) KMOSMO
SCHEMBL1317654 0.78 ACLY (0.62) ACLYHDAC1SUCNR1DHODH
SCHEMBL2275453 0.77 ACLY (0.76) ACLYHDAC1MEN1KMT2ASUCNR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7999132-B2 Anthranilic acid derivative or salt thereof TOYAMA CHEMICAL CO., LTD. (JP) 2011-08-16 US disclosed
US-20090240052-A1 NOVEL ANTHRANILIC ACID DERIVATIVE OR SALT THEREOF TOYAMA CHEMICAL CO., LTD. (JP) 2009-09-24 US disclosed
EP-1820795-A1 NOVEL ANTHRANILIC ACID DERIVATIVE OR SALT THEREOF TOYAMA CHEMICAL CO., LTD. (JP) 2007-08-22 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20090240052-A1 NOVEL ANTHRANILIC ACID DERIVATIVE OR SALT THEREOF MMP13, MMP26, MMP11 ACLY 653/4885KMO 194/4885HDAC1 71/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.