SCHEMBL22787828

SCHEMBL22787828

C=CCN([C@@H](C(=O)OC(C)(C)C)C(C)C)S(=O)(=O)c1ccc(OC)cc1

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.47
MEN1 O00255 3/20 0.47
MMP2 P08253 10/20 0.45
MMP9 P14780 10/20 0.45
MMP8 P22894 9/20 0.45
MMP13 P45452 9/20 0.45
KEAP1 Q14145 2/20 0.44
NFE2L2 Q16236 1/20 0.44
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
CA9 Q16790 1/20 0.43
ALOX12 P18054 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
BMP1 P13497 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14652641 0.83 MMP2 (0.47) MMP2MMP9MMP8MMP13KEAP1
SCHEMBL6076540 0.82 KEAP1 (0.41) MMP2MMP9MMP13KEAP1NFE2L2
SCHEMBL7089280 0.82 MMP2 (0.59) MMP2MMP9MMP8MMP13KEAP1
SCHEMBL7089279 0.82 MMP2 (0.59) MMP2MMP9MMP8MMP13KEAP1
SCHEMBL6498314 0.80 ADAMTS4 (0.47) KMT2AMEN1MMP2MMP9MMP8
SCHEMBL5451163 0.79 TAS2R14 (0.64) MMP2MMP9MMP8MMP13BMP1
SCHEMBL7387786 0.79 KEAP1 (0.38) MMP2MMP9MMP13KEAP1NFE2L2
SCHEMBL11956143 0.79 BMP1 (0.54) MMP2MMP9MMP8MMP13BMP1
SCHEMBL5463131 0.79 BMP1 (0.54) MMP2MMP9MMP8MMP13BMP1
SCHEMBL6388691 0.78 MMP2 (0.51) MMP2MMP9MMP8MMP13BMP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020252439-A1 CARBORANE HYDROXAMIC ACID MATRIX METALLOPROTEINASE AGENTS FOR BORON NEUTRON CAPTURE THERAPY LOYOLA UNIVERSITY OF CHICAGO (US) 2020-12-17 WO disclosed