SCHEMBL2280822

SCHEMBL2280822

Cc1cccc(C(C)(C)C)c1-c1[c]cccc1

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
GABRA1 P14867 1/20 0.43
GABRB2 P47870 1/20 0.43
CA2 P00918 1/20 0.35
ALDH1A1 P00352 3/20 0.34
TSHR P16473 2/20 0.34
TDP1 Q9NUW8 1/20 0.34
CYP2A6 P11509 2/20 0.31
CYP1A2 P05177 1/20 0.31
KIF11 P52732 1/20 0.31
GRIN2D O15399 1/20 0.30
GRIN3B O60391 1/20 0.30
GRIN1 Q05586 1/20 0.30
GRIN2A Q12879 1/20 0.30
GRIN2B Q13224 1/20 0.30
GRIN2C Q14957 1/20 0.30
GRIN3A Q8TCU5 1/20 0.30
SIGMAR1 Q99720 1/20 0.30
ACHE P22303 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28154136 0.89 CA2 (0.40) GABRA1GABRB2CA2ALDH1A1TSHR
SCHEMBL3223109 0.83 CYP1A2 (0.40) CA2ALDH1A1TSHRTDP1CYP2A6
SCHEMBL14877302 0.77 GABRA1 (0.60) GABRA1GABRB2CA2ALDH1A1TSHR
SCHEMBL445399 0.74 ALDH1A1 (0.39) GABRA1GABRB2CA2ALDH1A1TSHR
SCHEMBL2302604 0.74 TSHR (0.36) ALDH1A1TSHRTDP1CYP1A2
SCHEMBL2050623 0.72 CA2 (0.35) GABRA1GABRB2CA2ALDH1A1TSHR
SCHEMBL1160034 0.72 GABRA1 (0.50) GABRA1GABRB2CA2ALDH1A1TSHR
SCHEMBL29235924 0.72 GABRA1 (0.50) GABRA1GABRB2CA2ALDH1A1TSHR
SCHEMBL2280826 0.71 GABRA1 (0.46) GABRA1GABRB2CA2ALDH1A1TSHR
SCHEMBL499732 0.70 CA2 (0.31) CA2ALDH1A1TSHRTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110207956-A1 INTRAMOLECULAR C-H AMINATION WITH PHOSPHORYL AZIDES NATIONAL SCIENCE FOUNDATION 2011-08-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110207956-A1 INTRAMOLECULAR C-H AMINATION WITH PHOSPHORYL AZIDES CYCS, CCNH, CBR3 GABRA1 3242/4885GABRB2 3138/4885CA2 826/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.