SCHEMBL22809686

SCHEMBL22809686

Cc1cc(-n2ccc(N)nc2=O)cc(C)c1C

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 5/20 0.36
ADORA2A P29274 1/20 0.34
ADORA1 P30542 1/20 0.34
NOS3 P29474 1/20 0.33
NOS1 P29475 1/20 0.33
NOS2 P35228 1/20 0.33
LCK P06239 3/20 0.32
KIT P10721 3/20 0.32
SRC P12931 3/20 0.32
KDR P35968 1/20 0.32
BRPF1 P55201 1/20 0.32
COMT P21964 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
FGFR1 P11362 1/20 0.32
LMNA P02545 2/20 0.31
THRB P10828 1/20 0.31
MTOR P42345 1/20 0.31
MDM2 Q00987 1/20 0.31
NCOA1 Q15788 1/20 0.31
NCOA3 Q9Y6Q9 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24017805 0.85 HCAR1 (0.42) NOS3NOS1NOS2LCKKIT
SCHEMBL22386367 0.79 ALDH1A1 (0.42) ROCK2LCKKITSRCSMN1; SMN2
SCHEMBL22995728 0.79 XDH (0.42) ROCK2ADORA2ASMN1; SMN2LMNAALDH1A1
SCHEMBL22233947 0.79 NPC1 (0.43) ROCK2LCKKITSRCKDR
SCHEMBL20019313 0.79 MAT2A (0.39) LCKKITSRCSMN1; SMN2LMNA
SCHEMBL23678820 0.78 LCK (0.34) ROCK2NOS3NOS1NOS2LCK
SCHEMBL22386326 0.75 ROCK2 (0.39) ROCK2LCKSMN1; SMN2FGFR1LMNA
SCHEMBL2113288 0.75 SMN1; SMN2 (0.52) LCKKITSRCCOMTSMN1; SMN2
SCHEMBL22870491 0.75 XDH (0.40) NOS3NOS1NOS2COMT
SCHEMBL24285423 0.74 ELANE (0.41) ROCK2NOS3NOS2LCKKIT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3239134-B1 PYRIDONE AMIDES AS MODULATORS OF SODIUM CHANNELS VERTEX PHARMA (US) 2020-12-23 EP disclosed