SCHEMBL22852845

SCHEMBL22852845

COc1cc(F)ccc1Nc1cccc(C(F)(F)F)c1C(=O)O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.46
APAF1 O14727 1/20 0.46
RECQL P46063 1/20 0.46
CASP6 P55212 1/20 0.46
CACNA1B Q00975 1/20 0.46
APBA1 Q02410 1/20 0.46
MCL1 Q07820 1/20 0.46
CASP8 Q14790 1/20 0.46
SMO Q99835 1/20 0.46
FABP4 P15090 1/20 0.45
MAPK10 P53779 1/20 0.45
AKR1C3 P42330 3/20 0.44
AKR1C2 P52895 3/20 0.44
TAS2R14 Q9NYV8 2/20 0.43
RXFP1 Q9HBX9 1/20 0.43
CA12 O43570 1/20 0.43
CA1 P00915 1/20 0.43
CA2 P00918 1/20 0.43
CA7 P43166 1/20 0.43
CA9 Q16790 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30294776 1.00 KDM4E (0.46) KDM4EAPAF1RECQLCASP6CACNA1B
SCHEMBL30294255 0.85 ALDH1A1 (0.45) KDM4ESMOMAPK10RXFP1MAPT
SCHEMBL22853399 0.85 ALDH1A1 (0.45) KDM4ESMOMAPK10RXFP1MAPT
SCHEMBL30294602 0.84 TAS2R14 (0.49) FABP4AKR1C3AKR1C2TAS2R14ALDH1A1
SCHEMBL22852844 0.84 TAS2R14 (0.49) FABP4AKR1C3AKR1C2TAS2R14ALDH1A1
SCHEMBL22853486 0.80 MAPT (0.48) KDM4EMAPK10RXFP1MAPTSMN1; SMN2
SCHEMBL30294677 0.80 MAPT (0.48) KDM4EMAPK10RXFP1MAPTSMN1; SMN2
SCHEMBL20639015 0.79 SCN8A (0.47) CA12CA1CA2CA7CA9
SCHEMBL425534 0.77 CA12 (0.67) KDM4EAKR1C3AKR1C2CA12CA1
SCHEMBL22853079 0.76 MPO (0.57) KDM4EAPAF1RECQLCASP6CACNA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2020261114-A1 2,3-DIHYDROQUINAZOLIN COMPOUNDS AS NAV1.8 INHIBITORS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2020-12-30 WO disclosed