SCHEMBL22909452

SCHEMBL22909452

CN(C)Sc1c(F)c(F)c(F)c(F)c1CCc1ccc(C#N)cc1

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.38
NSD2 O96028 1/20 0.36
MAOA P21397 3/20 0.36
MAOB P27338 3/20 0.36
TSHR P16473 1/20 0.36
HSD17B10 Q99714 1/20 0.36
LOXL2 Q9Y4K0 2/20 0.36
KCNJ1 P48048 1/20 0.36
KCNH2 Q12809 1/20 0.36
HRH3 Q9Y5N1 3/20 0.35
DAO P14920 2/20 0.33
LSS P48449 1/20 0.33
IDO1 P14902 2/20 0.32
AR P10275 1/20 0.32
CYP19A1 P11511 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22909233 0.81 GFER (0.42) MAOAMAOBTSHRCYP19A1
SCHEMBL22909374 0.81 TAAR1 (0.39) TSHR
SCHEMBL22909268 0.78 ALDH1A1 (0.41) HSD17B10LOXL2HRH3
SCHEMBL22909382 0.72 SIGMAR1 (0.40) KCNH2
SCHEMBL10452241 0.71 LOXL2 (0.56) CYP2A6MAOAMAOBTSHRHSD17B10
SCHEMBL1004267 0.69 LOXL2 (0.64) CYP2A6MAOAMAOBTSHRHSD17B10
SCHEMBL22909581 0.68 DAO (0.37) MAOBKCNH2DAOIDO1
SCHEMBL22909469 0.67 ALDH1A1 (0.37) TSHR
SCHEMBL10924184 0.67 LSS (0.57) CYP2A6NSD2TSHRHSD17B10LOXL2
SCHEMBL10452156 0.66 TSHR (0.59) CYP2A6MAOAMAOBTSHRHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021009568-A1 BENZENESULFONAMIDE DERIVATIVES AND USES THEREOF 2692372 ONTARIO, INC. (CA) 2021-01-21 WO disclosed