SCHEMBL2295543

SCHEMBL2295543

CCCc1ccc(C2C(C(=O)c3ccc(C)cc3)C(O)=CN2CC(C)O)cc1

nearest known ligand 0.48

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ANXA2 P07355 6/20 0.48
S100A10 P60903 6/20 0.48
MGLL Q99685 1/20 0.33
PLK1 P53350 1/20 0.33
THRB P10828 2/20 0.32
ALDH1A1 P00352 2/20 0.32
L3MBTL1 Q9Y468 2/20 0.32
TDP1 Q9NUW8 2/20 0.32
LMNA P02545 1/20 0.32
ESR1 P03372 1/20 0.32
ESR2 Q92731 1/20 0.32
ENPP1 P22413 1/20 0.31
KCNH2 Q12809 1/20 0.31
CNR2 P34972 1/20 0.31
TAS1R3 Q7RTX0 1/20 0.31
TAS1R1 Q7RTX1 1/20 0.31
GAA P10253 1/20 0.31
THRA P10827 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2234747 0.86 L3MBTL1 (0.39) ANXA2S100A10MGLLALDH1A1L3MBTL1
SCHEMBL2234313 0.73 ANXA2 (0.45) ANXA2S100A10MGLLALDH1A1LMNA
SCHEMBL2295548 0.69 ANXA2 (0.55) ANXA2S100A10PLK1ALDH1A1L3MBTL1
SCHEMBL27449104 0.64 ALDH1A1 (0.64) PLK1THRBALDH1A1L3MBTL1TDP1
SCHEMBL14098923 0.61 KMT2A (0.61) PLK1THRBALDH1A1L3MBTL1LMNA
SCHEMBL19875785 0.60 PLK1 (0.47) PLK1THRBALDH1A1L3MBTL1TDP1
SCHEMBL19875784 0.60 PLK1 (0.47) PLK1THRBALDH1A1L3MBTL1TDP1
Hydrogen Peroxide SCHEMBL27723527 0.60 CYP1A2 (0.54) PLK1THRBALDH1A1L3MBTL1TDP1
SCHEMBL5493944 0.59 CYP1A2 (0.59) MGLLPLK1TDP1KCNH2CNR2
SCHEMBL326914 0.59 CYP1A2 (0.59) MGLLPLK1TDP1KCNH2CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011092505-A1 S100 PROTEIN BINDING INTERACTION INHIBITORS CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2011-08-04 WO claimed
WO-2011092505-A1 S100 PROTEIN BINDING INTERACTION INHIBITORS CANCER RESEARCH TECHNOLOGY LIMITED (GB) 2011-08-04 WO disclosed