SCHEMBL2302715

SCHEMBL2302715

NS(=O)(=O)c1ccc(N2CCNC2=O)cc1-c1cccc(Br)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 5/20 0.45
PTGS1 P23219 1/20 0.35
L3MBTL1 Q9Y468 2/20 0.34
CA1 P00915 4/20 0.34
CA2 P00918 4/20 0.34
CA9 Q16790 4/20 0.34
MMP2 P08253 2/20 0.34
MMP9 P14780 2/20 0.34
EIF2AK2 P19525 1/20 0.34
ALOX5AP P20292 1/20 0.34
FEN1 P39748 1/20 0.34
ALOX5 P09917 1/20 0.33
CA12 O43570 3/20 0.33
CA7 P43166 2/20 0.33
CA4 P22748 1/20 0.33
CA6 P23280 1/20 0.33
CA13 Q8N1Q1 1/20 0.33
CA5B Q9Y2D0 1/20 0.33
CA14 Q9ULX7 1/20 0.33
CDK2 P24941 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2301215 0.87 CA2 (0.37) PTGS2PTGS1CA1CA2CA9
SCHEMBL2299883 0.87 EIF2AK2 (0.41) PTGS2CA1CA2CA9EIF2AK2
SCHEMBL2303487 0.86 PTGS2 (0.45) PTGS2PTGS1ALOX5
SCHEMBL2301613 0.84 TGFBR1 (0.42) PTGS2CA1CA2CA9MMP2
SCHEMBL2300248 0.84 NISCH (0.37) MMP2ALOX5
SCHEMBL2302364 0.83 USP2 (0.36) CA1CA2EIF2AK2ALOX5
SCHEMBL2300517 0.81 PTGS2 (0.41) PTGS2PTGS1CA1CA2CA9
SCHEMBL2302290 0.81 ACVR1 (0.39) PTGS2PTGS1L3MBTL1CA1CA2
SCHEMBL2303196 0.81 PTGS2 (0.44) PTGS2PTGS1CA1CA2CA9
SCHEMBL2302226 0.80 CA1 (0.34) PTGS2CA1CA2CA9EIF2AK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2536693-A1 SUBSTITUTED 2-IMIDAZOLIDONES AND ANALOGS Université Laval (CA) 2012-12-26 EP disclosed
WO-2011100840-A1 SUBSTITUTED 2-IMIDAZOLIDONES AND ANALOGS UNIVERSITé LAVAL (CA) 2011-08-25 WO disclosed