SCHEMBL23146

SCHEMBL23146

COc1cc(C(=O)c2nc3ccccc3s2)c(OC)cc1C

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.53
MEN1 O00255 8/20 0.51
KMT2A Q03164 8/20 0.51
MAPT P10636 11/20 0.50
KDM4E B2RXH2 7/20 0.50
GAA P10253 4/20 0.50
HTT P42858 3/20 0.50
GLO1 Q04760 1/20 0.50
SMN1; SMN2 Q16637 5/20 0.49
TDP1 Q9NUW8 3/20 0.49
LMNA P02545 3/20 0.49
MAPK1 P28482 2/20 0.49
RECQL P46063 1/20 0.49
TP53 P04637 3/20 0.48
NPC1 O15118 4/20 0.48
KLF5 Q13887 1/20 0.48
BCL2 P10415 1/20 0.47
MCL1 Q07820 1/20 0.47
BAD Q92934 1/20 0.47
ATM Q13315 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30920 0.88 MAPT (0.56) ALDH1A1MEN1KMT2AMAPTKDM4E
SCHEMBL14021104 0.83 RAB9A (0.62) ALDH1A1MEN1KMT2AMAPTKDM4E
SCHEMBL28480483 0.78 ALDH1A1 (0.56) ALDH1A1MEN1KMT2AMAPTGAA
SCHEMBL427929 0.77 TUBB4A (0.72) ALDH1A1MEN1KMT2AMAPTKDM4E
SCHEMBL154083 0.74 ALDH1A1 (0.49) ALDH1A1MEN1KMT2AGLO1SMN1; SMN2
SCHEMBL6319718 0.74 ALDH1A1 (0.66) ALDH1A1MEN1KMT2AMAPTGAA
SCHEMBL31405 0.74 HSD17B1 (0.70) ALDH1A1MEN1KMT2AMAPTKDM4E
SCHEMBL8405393 0.72 MAOB (0.64) ALDH1A1MEN1KMT2AKDM4EHTT
SCHEMBL13833752 0.72 ALDH1A1 (0.53) ALDH1A1MEN1KMT2AMAPTKDM4E
SCHEMBL11007700 0.72 KMT2A (0.66) ALDH1A1MEN1KMT2AMAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2609089-A1 SELECTIVE 17BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 INHIBITORS Universität des Saarlandes (DE) 2013-07-03 EP disclosed
WO-2012025638-A1 SELECTIVE 17BETA-HYDROXYSTEROID DEHYDROGENASE TYPE 1 INHIBITORS Universität des Saarlandes (DE) 2012-03-01 WO disclosed