Berberine

Berberine

SCHEMBL231931

COc1ccc2cc3[n+](cc2c1OC)CCc1cc2c(cc1-3)OCO2.[N-]=[N+]=[N-]

nearest known ligand 0.92

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 10/20 0.92
BCHE P06276 9/20 0.92
EP300 Q09472 5/20 0.92
LMNA P02545 3/20 0.92
CYP3A4 P08684 3/20 0.92
CYP2D6 P10635 3/20 0.92
MAPT P10636 3/20 0.92
RAD52 P43351 3/20 0.92
ALDH1A1 P00352 2/20 0.92
CHRM1 P11229 2/20 0.92
DRD2 P14416 2/20 0.92
TSHR P16473 2/20 0.92
ADRA2B P18089 2/20 0.92
ADRA2C P18825 2/20 0.92
RXRA P19793 2/20 0.92
DRD1 P21728 2/20 0.92
HTR2B P41595 2/20 0.92
HTT P42858 2/20 0.92
KCNH2 Q12809 2/20 0.92
SMN1; SMN2 Q16637 2/20 0.92

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Berberine SCHEMBL29354144 0.96 ACHE (1.00) ACHEBCHEEP300LMNACYP3A4
Berberine SCHEMBL15669190 0.96 ACHE (1.00) ACHEBCHEEP300LMNACYP3A4
Berberine SCHEMBL25632 0.96 ACHE (1.00) ACHEBCHEEP300LMNACYP3A4
Berberine SCHEMBL30153843 0.96 ACHE (1.00) ACHEBCHEEP300LMNACYP3A4
Berberine SCHEMBL4894622 0.95 BCHE (0.98) ACHEBCHEEP300LMNACYP3A4
Berberine SCHEMBL1376273 0.95 ACHE (0.98) ACHEBCHEEP300LMNACYP3A4
Berberine SCHEMBL3686644 0.95 ACHE (0.98) ACHEBCHEEP300LMNACYP3A4
Berberine SCHEMBL21462194 0.95 ACHE (0.98) ACHEBCHEEP300LMNACYP3A4
Berberine SCHEMBL153906 0.95 ACHE (1.00) ACHEBCHEEP300LMNACYP3A4
Berberine SCHEMBL2538316 0.95 ACHE (0.98) ACHEBCHEEP300LMNACYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 35 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2361625-A1 Methods and compositions for the treatment of hyperlipidemia Institute of Medicinal Biotechnology, Chinese Academy of Medical Sciences (CN) 2011-08-31 EP claimed
US-20110158932-A1 Methods And Compositions For The Treatment of Hyperlipidemia ABBOTT LABORATORIES 2011-06-30 US claimed
EP-1796666-A4 METHODS AND COMPOSITIONS FOR THE TREATMENT OF HYPERLIPIDEMIA INST MEDICINAL BIOTECHNOLOGY (CN) 2008-03-19 EP claimed
CN-101102768-A Method and composition for the treatment of hyperlipidemia MEDICINE AND BIOENGINEERING IN (CN) 2008-01-09 CN claimed
EP-1796666-A1 METHODS AND COMPOSITIONS FOR THE TREATMENT OF HYPERLIPIDEMIA Institute of Medicinal Biotechnology, Chinese Acadamy of Medical Sciences (CN) 2007-06-20 EP claimed
US-20060223838-A1 Methods and compositions for the treatment of hyperlipidemia INSTITUTE OF MEDICINAL BIOTECHNOLOGY (CN) 2006-10-05 US claimed
WO-2006029577-A9 METHODS AND COMPOSITIONS FOR THE TREATMENT OF HYPERLIPIDEMIA INST MEDICINAL BIOTECHNOLOGY (CN) 2006-05-26 WO claimed
WO-2006029577-A1 METHODS AND COMPOSITIONS FOR THE TREATMENT OF HYPERLIPIDEMIA INSTITUTE OF MEDICINAL BIOTECHNOLOGY, CHINESE ACADEMY OF MEDICAL SCIENCES (CN) 2006-03-23 WO claimed
US-20220387403-A1 COMPOUNDS, COMPOSITIONS AND METHODS FOR TREATING NASH, NAFLD, AND OBESITY CVI PHARMACEUTICALS LIMITED (KY) 2022-12-08 US disclosed
WO-2021067490-A1 COMPOUNDS, COMPOSITIONS AND METHODS FOR TREATING NASH, NAFLD, AND OBESITY CVI PHARMACEUTICALS LIMITED (KY) 2021-04-08 WO disclosed
CN-105777632-A Aromatic-ring azacyclo derivatives and application thereof 成都贝斯凯瑞生物科技有限公司 2016-07-20 CN disclosed
CN-105777633-A Tetrahydroisoquinoline derivative and application thereof 成都贝斯凯瑞生物科技有限公司 2016-07-20 CN disclosed
CN-105753817-A Nitrogen-substituted heterocyclic derivatives and application thereof 成都贝斯凯瑞生物科技有限公司 2016-07-13 CN disclosed
CN-105753814-A Substituted nitrogen heterocyclic derivative and application thereof 成都贝斯凯瑞生物科技有限公司 2016-07-13 CN disclosed
EP-1796666-A4 METHODS AND COMPOSITIONS FOR THE TREATMENT OF HYPERLIPIDEMIA INST MEDICINAL BIOTECHNOLOGY (CN) 2008-03-19 EP disclosed
CN-101102768-A Method and composition for the treatment of hyperlipidemia MEDICINE AND BIOENGINEERING IN (CN) 2008-01-09 CN disclosed
EP-1796666-A1 METHODS AND COMPOSITIONS FOR THE TREATMENT OF HYPERLIPIDEMIA Institute of Medicinal Biotechnology, Chinese Acadamy of Medical Sciences (CN) 2007-06-20 EP disclosed
US-20060223838-A1 Methods and compositions for the treatment of hyperlipidemia INSTITUTE OF MEDICINAL BIOTECHNOLOGY (CN) 2006-10-05 US disclosed
WO-2006029577-A9 METHODS AND COMPOSITIONS FOR THE TREATMENT OF HYPERLIPIDEMIA INST MEDICINAL BIOTECHNOLOGY (CN) 2006-05-26 WO disclosed
WO-2006029577-A1 METHODS AND COMPOSITIONS FOR THE TREATMENT OF HYPERLIPIDEMIA INSTITUTE OF MEDICINAL BIOTECHNOLOGY, CHINESE ACADEMY OF MEDICAL SCIENCES (CN) 2006-03-23 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20220387403-A1 COMPOUNDS, COMPOSITIONS AND METHODS FOR TREATING NASH, NAFLD, AND OBESITY LIPC, FABP1, CPT1A ACHE 2228/4885BCHE 795/4885EP300 212/4885
US-20110158932-A1 Methods And Compositions For The Treatment of Hyperlipidemia PCSK9, APOB, LDLR ACHE 69/4885BCHE 33/4885EP300 3709/4885
US-20060223838-A1 Methods and compositions for the treatment of hyperlipidemia PCSK9, APOB, LDLR ACHE 69/4885BCHE 33/4885EP300 3709/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.