SCHEMBL23201480

SCHEMBL23201480

CC(C)c1nccc(CO[Si](c2ccccc2)(c2ccccc2)C(C)(C)C)c1N

nearest known ligand 0.40

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
SMYD2 Q9NRG4 2/20 0.33
POLB P06746 1/20 0.32
CYP3A4 P08684 1/20 0.30
HTT P42858 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
DHFR P00374 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23234695 0.80 FFAR2 (0.31) SMYD2CYP3A4HTTSMN1; SMN2
SCHEMBL21543198 0.80 SLC16A3 (0.32) SMYD2CYP3A4HTTSMN1; SMN2
SCHEMBL2598798 0.75 LTA4H (0.41) SMYD2HTTSMN1; SMN2
SCHEMBL21639770 0.74 AOC1 (0.45)
SCHEMBL21543547 0.74 IDO1 (0.38) HTT
SCHEMBL4298877 0.71 NOS3 (0.45) SMYD2
SCHEMBL4821504 0.71 SMYD2 (0.33) SMYD2CYP3A4HTTSMN1; SMN2
SCHEMBL3598198 0.70 ALOX5AP (0.41) SMYD2CYP3A4HTTSMN1; SMN2DHFR
SCHEMBL23272953 0.70 DUT (0.30)
SCHEMBL29823172 0.70 DUT (0.30)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12583854-B2 KRAS G12C inhibitors and methods of using the same AMGEN INC. (US) 2026-03-24 US disclosed
US-12083121-B2 Substituted piperazines as KRAS G12C inhibitors AMGEN INC. (US) 2024-09-10 US disclosed
EP-4268898-A2 KRAS G12C INHIBITORS FOR TREATING CANCER Amgen Inc. (US) 2023-11-01 EP disclosed
US-20220175782-A1 KRAS G12C INHIBITORS AND METHODS OF USING THE SAME AMGEN INC. 2022-06-09 US disclosed
US-11285156-B2 Substituted piperazines as KRAS G12C inhibitors AMGEN INC. (US) 2022-03-29 US disclosed
US-20220002298-A1 KRAS G12C INHIBITORS AND METHODS OF USING THE SAME AMGEN INC. 2022-01-06 US disclosed
EP-3807276-A2 KRAS G12C INHIBITORS ENCOMPASSING A PIPERAZINE RING AND USE THEREOF IN THE TREATMENT OF CANCER Amgen Inc. (US) 2021-04-21 EP disclosed
EP-3802537-A1 KRAS G12C INHIBITORS FOR TREATING CANCER Amgen Inc. (US) 2021-04-14 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11285156-B2 Substituted piperazines as KRAS G12C inhibitors KRAS, NRAS, HRAS SMYD2 1861/4885POLB 596/4885CYP3A4 4426/4885
US-12083121-B2 Substituted piperazines as KRAS G12C inhibitors KRAS, NRAS, HRAS SMYD2 1861/4885POLB 596/4885CYP3A4 4426/4885
US-12583854-B2 KRAS G12C inhibitors and methods of using the same KRAS, NRAS, APC SMYD2 684/4885POLB 2374/4885CYP3A4 4767/4885
US-20220175782-A1 KRAS G12C INHIBITORS AND METHODS OF USING THE SAME KRAS, NRAS, HRAS SMYD2 1431/4885POLB 632/4885CYP3A4 4763/4885
US-20220002298-A1 KRAS G12C INHIBITORS AND METHODS OF USING THE SAME KRAS, NRAS, HRAS SMYD2 1431/4885POLB 632/4885CYP3A4 4763/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.