SCHEMBL232086

SCHEMBL232086

N#Cc1ccc(N2CCNCC2)c(F)c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.57
DRD2 P14416 1/20 0.53
DRD3 P35462 1/20 0.53
MAPKAPK2 P49137 1/20 0.45
SLC6A9 P48067 5/20 0.45
ADRA1D P25100 1/20 0.45
ADRA1A P35348 1/20 0.45
ADRA1B P35368 1/20 0.45
SLC6A5 Q9Y345 2/20 0.43
HTR6 P50406 1/20 0.42
ADRB1 P08588 1/20 0.42
MAPT P10636 2/20 0.42
KDM4E B2RXH2 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
OPRL1 P41146 1/20 0.42
HRH4 Q9H3N8 1/20 0.42
HRH3 Q9Y5N1 1/20 0.42
KDR P35968 1/20 0.41
LMNA P02545 1/20 0.41
GAA P10253 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29380294 1.00 ALDH1A1 (0.57) ALDH1A1DRD2DRD3MAPKAPK2SLC6A9
Hydrochloric Acid SCHEMBL22532864 0.98 ALDH1A1 (0.56) ALDH1A1DRD2DRD3MAPKAPK2SLC6A9
Hydrochloric Acid SCHEMBL29380273 0.98 ALDH1A1 (0.56) ALDH1A1DRD2DRD3MAPKAPK2SLC6A9
Hydrochloric Acid SCHEMBL29882265 0.98 ALDH1A1 (0.56) ALDH1A1DRD2DRD3MAPKAPK2SLC6A9
SCHEMBL25629584 0.94 ALDH1A1 (0.52) ALDH1A1DRD2DRD3MAPKAPK2SLC6A9
Hydrochloric Acid SCHEMBL31720538 0.93 ALDH1A1 (0.51) ALDH1A1DRD2DRD3MAPKAPK2SLC6A9
SCHEMBL3164773 0.87 ALDH1A1 (0.57) ALDH1A1DRD2DRD3MAPKAPK2HTR6
Hydrochloric Acid SCHEMBL23303687 0.85 ALDH1A1 (0.56) ALDH1A1DRD2DRD3MAPKAPK2HTR6
SCHEMBL15117102 0.85 SLC6A9 (0.57) ALDH1A1SLC6A9ADRA1DADRA1AADRA1B
SCHEMBL8415671 0.82 SLC6A9 (0.46) ALDH1A1SLC6A9ADRA1DADRA1AADRA1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 230 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4467143-B1 METHOD FOR PREPARING 4-(4-(4-(((2-(2,6-DIOXOPIPERIDIN-3-YL)-L-OXOISOINDOLIN-4-YL)OXY)METHYL)BENZYL)PIPERAZIN-L-YL)-3-FLUOROBENZONITRILE CELGENE CORP (US) 2026-03-11 EP claimed
EP-4467143-A2 4-(4-(4-(((2-(2,6-DIOXOPIPERIDIN-3-YL)-L-OXOISOINDOLIN-4-YL)OXY)METHYL)BENZYL)PIPERAZIN-L-YL)-3-FLUOROBENZONITRILE AS ANTIPROLIFERATIVE COMPOUND Celgene Corporation (US) 2024-11-27 EP claimed
US-12029738-B2 Antiproliferative compounds and methods of use thereof CELGENE CORPORATION (US) 2024-07-09 US claimed
US-20220280505-A1 ANTIPROLIFERATIVE COMPOUNDS AND METHODS OF USE THEREOF CELGENE CORPORATION 2022-09-08 US claimed
US-10675281-B2 Antiproliferative compounds and methods of use thereof CELGENE CORPORATION (US) 2020-06-09 US claimed
EP-4100410-B1 MUSCARINIC RECEPTOR 4 ANTAGONISTS AND METHODS OF USE NEUROCRINE BIOSCIENCES INC (US) 2026-04-22 EP disclosed
EP-4725553-A2 SOLID FORMS COMPRISING (S)-4-(4-(4-(((2-(2,6-DIOXOPIPERIDIN-3-YL)-1-OXOISOINDOLIN-4-YL)OXY)METHYL) BENZYL)PIPERAZIN-1-YL)-3-FLUOROBENZONITRILE AND SALTS THEREOF, AND COMPOSITIONS COMPRISING AND METHODS OF USING THE SAME Celgene Corporation (US) 2026-04-15 EP disclosed
US-12582641-B2 Sulfur-containing compound based on glutarimide skeleton and application thereof SHANGHAITECH UNIVERSITY (CN) 2026-03-24 US disclosed
EP-4467143-B1 METHOD FOR PREPARING 4-(4-(4-(((2-(2,6-DIOXOPIPERIDIN-3-YL)-L-OXOISOINDOLIN-4-YL)OXY)METHYL)BENZYL)PIPERAZIN-L-YL)-3-FLUOROBENZONITRILE CELGENE CORP (US) 2026-03-11 EP disclosed
US-20260001863-A1 NOVEL PYRIDAZINES BOEHRINGER INGELHEIM INT (DE) 2026-01-01 US disclosed
US-12510533-B2 Methods for treating multiple myeloma and the use of companion biomarkers for 4-(4-(4-(((2-(2,6-dioxopiperidin-3-yl)-1-oxoisoindolin-4-yl)oxy)methyl)benzyl)piperazin-1-yl)-3-fluorobenzonitrile CELGENE CORPORATION (US) 2025-12-30 US disclosed
EP-3908582-B1 SOLID FORMS COMPRISING (S)-4-(4-(4-(((2-(2,6-DIOXOPIPERIDIN-3-YL)-1-OXOISOINDOLIN-4-YL)OXY)METHYL) BENZYL)PIPERAZIN-1-YL)-3-FLUOROBENZONITRILE AND SALTS THEREOF, AND COMPOSITIONS COMPRISING AND METHODS OF USING THE SAME CELGENE CORP (US) 2025-11-12 EP disclosed
US-6630475-B2 5-amino-pyrazolo-(4, 3-e)-1,2,4-triazolo(1,5-c)pyrimidine adenosine A2a receptor antagonists; use in the treatment of central nervous system diseases, in particular Parkinson's disease SCHERING CORPORATION 2003-10-07 US disclosed
EP-1283839-A1 ADENOSINE A2A RECEPTOR ANTAGONISTS SCHERING CORPORATION (US) 2003-02-19 EP disclosed
US-20020099061-A1 Adenosine A2a receptor antagonists MERCK SHARP & DOHME CORP. 2002-07-25 US disclosed
WO-2001092264-A1 ADENOSINE A2A RECEPTOR ANTAGONISTS SCHERING CORPORATION (US) 2001-12-06 WO disclosed
US-6013654-A Imidazo[1,2-A]pyridines for the treatment of CNS and cardiac diseases PHARMACIA & UPJOHN COMPANY (US) 2000-01-11 US disclosed
US-5912246-A Imidazo 1,2-a!pyridines for the treatment of CNS and cardiac diseases PHARMACIA & UPJOHN COMPANY (US) 1999-06-15 US disclosed
EP-0809642-A1 IMIDAZO 1,2-A]PYRIDINES FOR THE TREATMENT OF CNS AND CARDIAC DISEASES PHARMACIA & UPJOHN COMPANY (US) 1997-12-03 EP disclosed
WO-1996025414-A1 IMIDAZO[1,2-A]PYRIDINES FOR THE TREATMENT OF CNS AND CARDIAC DISEASES PHARMACIA & UPJOHN COMPANY (US) 1996-08-22 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-12582641-B2 Sulfur-containing compound based on glutarimide skeleton and application thereof SUCNR1, SRD5A1, GLS ALDH1A1 697/4885DRD2 4186/4885DRD3 3575/4885
US-12029738-B2 Antiproliferative compounds and methods of use thereof MCL1, NPM1, NFATC1 ALDH1A1 2344/4885DRD2 4810/4885DRD3 4675/4885
US-10675281-B2 Antiproliferative compounds and methods of use thereof MCL1, NPM1, NFATC1 ALDH1A1 2344/4885DRD2 4810/4885DRD3 4675/4885
US-20260001863-A1 NOVEL PYRIDAZINES ENPP2, LPAR5, LPAR1 ALDH1A1 2616/4885DRD2 2576/4885DRD3 3251/4885
US-12510533-B2 Methods for treating multiple myeloma and the use of companion biomarkers for 4-(4-(4-(((2-(2,6-dioxopiperidin-3-yl)-1-oxoisoindolin-4-yl)oxy)methyl)benzyl)piperazin-1-yl)-3-fluorobenzonitrile IKZF1, IKZF3, IKZF2 ALDH1A1 3404/4885DRD2 4207/4885DRD3 3122/4885
US-20020099061-A1 Adenosine A2a receptor antagonists ADORA2A, ADORA3, ADORA2B ALDH1A1 2158/4885DRD2 75/4885DRD3 123/4885
US-20220280505-A1 ANTIPROLIFERATIVE COMPOUNDS AND METHODS OF USE THEREOF MCL1, NPM1, NFATC1 ALDH1A1 2344/4885DRD2 4810/4885DRD3 4675/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.