SCHEMBL23257562

SCHEMBL23257562

C=CC(=O)Nc1cc(C(=O)NCCc2cccc3ccc(OC)cc23)cc(C(F)(F)F)c1

nearest known ligand 0.61

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
TRPV1 Q8NER1 2/20 0.61
MTNR1A P48039 15/20 0.59
MTNR1B P49286 7/20 0.59
NQO2 P16083 3/20 0.59
HTR2C P28335 1/20 0.53
HTR2B P41595 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23256738 0.84 CA1 (0.52) MTNR1AMTNR1B
SCHEMBL9490469 0.83 MTNR1A (0.75) TRPV1MTNR1AMTNR1BNQO2HTR2C
SCHEMBL7017220 0.76 MTNR1A (1.00) TRPV1MTNR1AMTNR1BNQO2HTR2C
SCHEMBL9424922 0.75 MTNR1A (1.00) TRPV1MTNR1AMTNR1BNQO2HTR2C
SCHEMBL9493664 0.75 MTNR1A (0.81) TRPV1MTNR1AMTNR1BNQO2HTR2C
SCHEMBL9491217 0.73 MTNR1A (0.81) TRPV1MTNR1AMTNR1BNQO2HTR2C
SCHEMBL23257559 0.73 TGM2 (0.43)
SCHEMBL23257556 0.72 TGM2 (0.50)
SCHEMBL23256741 0.72 MEN1 (0.57)
Agomelatine SCHEMBL15822116 0.71 MTNR1A (0.84) TRPV1MTNR1AMTNR1BNQO2HTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021076755-A1 AN ACTIVITY-GUIDE MAP OF ELECTROPHILE-CYSTEINE INTERACTIONS IN PRIMARY HUMAN IMMUNE CELLS THE SCRIPPS RESEARCH INSTITUTE (US) 2021-04-22 WO disclosed