SCHEMBL2326348

SCHEMBL2326348

COC(=O)/C=C(\C)NC(C)=O

nearest known ligand 0.50

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.50
TSHR P16473 2/20 0.47
HCAR2 Q8TDS4 2/20 0.43
KEAP1 Q14145 1/20 0.43
NFE2L2 Q16236 1/20 0.43
ALDH1A1 P00352 4/20 0.36
CRBN Q96SW2 1/20 0.36
TAS2R38 P59533 1/20 0.33
ALOX15 P16050 1/20 0.31
RECQL P46063 1/20 0.31
HSD17B10 Q99714 1/20 0.31
KDM4E B2RXH2 2/20 0.31
MAPT P10636 1/20 0.31
TDP1 Q9NUW8 1/20 0.31
CA2 P00918 1/20 0.30
PTGS1 P23219 1/20 0.30
MMP12 P39900 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2326353 1.00 SMN1; SMN2 (0.50) SMN1; SMN2TSHRHCAR2KEAP1NFE2L2
SCHEMBL2326345 1.00 SMN1; SMN2 (0.50) SMN1; SMN2TSHRHCAR2KEAP1NFE2L2
SCHEMBL5143661 0.78 NPSR1 (0.50) SMN1; SMN2TSHRHCAR2ALDH1A1ALOX15
SCHEMBL12213573 0.78 NPSR1 (0.50) SMN1; SMN2TSHRHCAR2ALDH1A1ALOX15
SCHEMBL5143663 0.78 NPSR1 (0.50) SMN1; SMN2TSHRHCAR2ALDH1A1ALOX15
SCHEMBL11707587 0.77
SCHEMBL11708371 0.77 HCAR2 (0.46) SMN1; SMN2TSHRHCAR2KEAP1NFE2L2
SCHEMBL1739 0.77
SCHEMBL1740 0.77
SCHEMBL12431015 0.77

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012176830-A1 1,2-BIS(DIALKYLPHOSPHINO)-4,5-(METHYLENEDIOXY)BENZENE DERIVATIVE, METHOD FOR MANUFACTURING SAME, METAL COMPLEX HAVING THIS 1,2-BIS(DIALKYLPHOSPHINO)-4,5-(METHYLENEDIOXY)BENZENE DERIVATIVE AS A LIGAND, AND ASYMMETRIC HYDROGENATION METHOD 日本化学工業株式会社 (JP) 2012-12-27 WO disclosed
EP-2534161-A1 ENANTIOMERICALLY ENRICHED AMINODIPHOSPHINES AS LIGANDS FOR THE PREPARATION OF CATALYSTS FOR ASYMMETRIC SYNTHESIS Enantia, S.L. (ES) 2012-12-19 EP disclosed
US-20120309997-A1 Enantiomerically Enriched Aminodiphosphines as Ligands for the Preparation of Catalysts for Asymmetric Synthesis ENANTIA, S.L. (ES) 2012-12-06 US disclosed
US-20120309997-A1 Enantiomerically Enriched Aminodiphosphines as Ligands for the Preparation of Catalysts for Asymmetric Synthesis ENANTIA, S.L. (ES) 2012-12-06 US disclosed
WO-2011098160-A1 ENANTIOMERICALLY ENRICHED AMINODIPHOSPHINES AS LIGANDS FOR THE PREPARATION OF CATALYSTS FOR ASYMMETRIC SYNTHESIS ENANTIA, S.L. (ES) 2011-08-18 WO disclosed
WO-2011098160-A1 ENANTIOMERICALLY ENRICHED AMINODIPHOSPHINES AS LIGANDS FOR THE PREPARATION OF CATALYSTS FOR ASYMMETRIC SYNTHESIS ENANTIA, S.L. (ES) 2011-08-18 WO disclosed
US-20070197799-A1 Novel bisphosphane catalysts DEGUSSA GMBH (DE) 2007-08-23 US disclosed
US-20060183930-A1 Chiral monophosphorus compounds DREISBACH CLAUS 2006-08-17 US disclosed
US-7057061-B2 Chiral monophosphorus compounds BAYER AKTIENGESELLSCHAFT (DE) 2006-06-06 US disclosed
US-20030119664-A1 Chiral monophosphorus compounds LANXESS DEUTSCHLAND GMBH (DE) 2003-06-26 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070197799-A1 Novel bisphosphane catalysts BPGM, BCAT2, BCAT1 SMN1; SMN2 3430/4885TSHR 3358/4885HCAR2 3651/4885
US-20120309997-A1 Enantiomerically Enriched Aminodiphosphines as Ligands for the Preparation of Catalysts for Asymmetric Synthesis PHOSPHO1, AASDHPPT, AGPS SMN1; SMN2 4541/4885TSHR 4609/4885HCAR2 4276/4885
US-20060183930-A1 Chiral monophosphorus compounds PNP, MTAP, MDM4 SMN1; SMN2 4415/4885TSHR 4870/4885HCAR2 4736/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.