SCHEMBL23301686

SCHEMBL23301686

CS(=O)(=O)CCCn1c(C(=O)O)cc2cc(Cl)ccc21

nearest known ligand 0.55

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 15/20 0.55
MCL1 Q07820 2/20 0.45
ACLY P53396 1/20 0.45
ABCB11 O95342 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6750603 0.90 CCR9 (0.54) CCR2MCL1
SCHEMBL15416321 0.85 NOD2 (0.47) CCR2
SCHEMBL4372812 0.84 CCR2 (0.60) CCR2MCL1ABCB11
SCHEMBL23330647 0.82 ACLY (0.41) CCR2ACLY
SCHEMBL15685313 0.82 TDP1 (0.41) CCR2
SCHEMBL6750553 0.82 CCR9 (0.56) CCR2
SCHEMBL15416658 0.82 ACLY (0.47) CCR2ACLY
SCHEMBL16235858 0.82 CCR2 (0.59) CCR2MCL1ABCB11
SCHEMBL16235848 0.82 NOD2 (0.46) CCR2
SCHEMBL8687383 0.81 CCR2 (0.62) CCR2ABCB11

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240109894-A1 SYNTHESIS OF 3-({5-CHLORO-1-[3-(METHYLSULFONYL)PROPYL]-1H-INDOL-2-YL} METHYL)-1-(2,2,2-TRIFLUOROETHYL)-1,3-DIHYDRO-2H-IMIDAZO[4,5-C]PYRIDIN-2-ONE JOHNSON & JOHNSON (CHINA) INVESTMENT LTD. (CN) 2024-04-04 US claimed
EP-4051662-B1 SYNTHESIS OF 3-({5-CHLORO-1-[3-(METHYLSULFONYL)PROPYL]-1H-INDOL-2 YL}METHYL)-1-(2,2,2-TRIFLUOROETHYL)-1,3-DIHYDRO-2H-IMIDAZO[4,5-C]PYRIDIN-2-ONE JANSSEN SCIENCES IRELAND UNLIMITED CO (IE) 2024-02-07 EP claimed
CN-114630828-B Synthesis of RSV inhibition compound 杨森科学爱尔兰无限公司 2023-10-31 CN claimed
CN-114630828-A Synthesis of 3- ({ 5-chloro-1- [3- (methylsulfonyl) propyl ] -1H-indol-2-yl } methyl) -1- (2,2, 2-trifluoroethyl) -1, 3-dihydro-2H-imidazo [4,5-c ] pyridin-2-one 杨森科学爱尔兰无限公司 2022-06-14 CN claimed
WO-2021083998-A1 SYNTHESIS OF 3-({5-CHLORO-1-[3-(METHYLSULFONYL)PROPYL]-1H-INDOL-2 YL} METHYL)-1-(2,2,2-TRIFLUOROETHYL)-1,3-DIHYDRO-2H-IMIDAZO[4,5-C]PYRIDIN-2-ONE Janssen Sciences Ireland Unlimited Company (IE) 2021-05-06 WO claimed
US-20240109894-A1 SYNTHESIS OF 3-({5-CHLORO-1-[3-(METHYLSULFONYL)PROPYL]-1H-INDOL-2-YL} METHYL)-1-(2,2,2-TRIFLUOROETHYL)-1,3-DIHYDRO-2H-IMIDAZO[4,5-C]PYRIDIN-2-ONE JOHNSON & JOHNSON (CHINA) INVESTMENT LTD. (CN) 2024-04-04 US disclosed
EP-4051662-B1 SYNTHESIS OF 3-({5-CHLORO-1-[3-(METHYLSULFONYL)PROPYL]-1H-INDOL-2 YL}METHYL)-1-(2,2,2-TRIFLUOROETHYL)-1,3-DIHYDRO-2H-IMIDAZO[4,5-C]PYRIDIN-2-ONE JANSSEN SCIENCES IRELAND UNLIMITED CO (IE) 2024-02-07 EP disclosed
CN-114630828-B Synthesis of RSV inhibition compound 杨森科学爱尔兰无限公司 2023-10-31 CN disclosed
CN-114630828-A Synthesis of 3- ({ 5-chloro-1- [3- (methylsulfonyl) propyl ] -1H-indol-2-yl } methyl) -1- (2,2, 2-trifluoroethyl) -1, 3-dihydro-2H-imidazo [4,5-c ] pyridin-2-one 杨森科学爱尔兰无限公司 2022-06-14 CN disclosed
WO-2021083998-A1 SYNTHESIS OF 3-({5-CHLORO-1-[3-(METHYLSULFONYL)PROPYL]-1H-INDOL-2 YL} METHYL)-1-(2,2,2-TRIFLUOROETHYL)-1,3-DIHYDRO-2H-IMIDAZO[4,5-C]PYRIDIN-2-ONE Janssen Sciences Ireland Unlimited Company (IE) 2021-05-06 WO disclosed
WO-2021083998-A1 SYNTHESIS OF 3-({5-CHLORO-1-[3-(METHYLSULFONYL)PROPYL]-1H-INDOL-2 YL} METHYL)-1-(2,2,2-TRIFLUOROETHYL)-1,3-DIHYDRO-2H-IMIDAZO[4,5-C]PYRIDIN-2-ONE Janssen Sciences Ireland Unlimited Company (IE) 2021-05-06 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240109894-A1 SYNTHESIS OF 3-({5-CHLORO-1-[3-(METHYLSULFONYL)PROPYL]-1H-INDOL-2-YL} METHYL)-1-(2,2,2-TRIFLUOROETHYL)-1,3-DIHYDRO-2H-IMIDAZO[4,5-C]PYRIDIN-2-ONE HTR3C, MECP2, CDK2 CCR2 501/4885MCL1 1795/4885ACLY 3884/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.