SCHEMBL23372155

SCHEMBL23372155

CCc1c(N)ccc(C)c1F

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 1/20 0.39
NOS2 P35228 1/20 0.39
S100B P04271 1/20 0.38
KDM4E B2RXH2 1/20 0.34
POLB P06746 1/20 0.34
CYP3A4 P08684 5/20 0.33
TDP1 Q9NUW8 4/20 0.33
ALDH1A1 P00352 3/20 0.33
TSHR P16473 2/20 0.33
CASP1 P29466 1/20 0.33
SKP2 Q13309 1/20 0.33
ESR1 P03372 1/20 0.31
AR P10275 1/20 0.31
ESR2 Q92731 1/20 0.31
HTR2A P28223 1/20 0.30
HTR2C P28335 1/20 0.30
HTR2B P41595 1/20 0.30
TP53 P04637 1/20 0.30
THRB P10828 1/20 0.30
ALOX15 P16050 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24620497 0.86 NOS3 (0.35) NOS3NOS2S100BKDM4EPOLB
SCHEMBL25531700 0.84 NOS2 (0.45) NOS3NOS2S100BKDM4EPOLB
SCHEMBL11891674 0.81 NOS3 (0.40) NOS3NOS2KDM4EPOLBHTR2A
SCHEMBL6652156 0.80 ALDH1A1 (0.34) NOS3NOS2S100BKDM4EPOLB
SCHEMBL109396 0.79 NOS2 (0.48) NOS3NOS2S100BKDM4EPOLB
SCHEMBL2954428 0.77 NOS2 (0.42) NOS3NOS2S100BKDM4EPOLB
SCHEMBL6356384 0.77 NOS3 (0.42) NOS3NOS2S100BKDM4EPOLB
SCHEMBL12886698 0.77 ACHE (0.33) NOS3NOS2
SCHEMBL20079594 0.77 CYP3A4 (0.33) NOS3NOS2CYP3A4ALDH1A1TSHR
SCHEMBL15133727 0.76 P2RX7 (0.34) NOS3NOS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021096948-A1 ALLOSTERIC EGFR INHIBITORS AND METHODS OF USE THEREOF DANA-FARBER CANCER INSTITUTE, INC. (US) 2021-05-20 WO disclosed