SCHEMBL2340169

SCHEMBL2340169

COC(=O)c1ccc(CO[Si](C)(C)C(C)(C)C)[nH]1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 3/20 0.42
KDM4E B2RXH2 1/20 0.42
GLA P06280 1/20 0.42
BACE1 P56817 1/20 0.36
MMP2 P08253 1/20 0.35
DUT P33316 2/20 0.34
MAPK1 P28482 1/20 0.33
CYP1A2 P05177 1/20 0.33
LMNA P02545 2/20 0.32
ALDH1A1 P00352 1/20 0.32
RAB9A P51151 3/20 0.31
MAPT P10636 2/20 0.31
ALPL P05186 1/20 0.31
POLB P06746 1/20 0.31
CA12 O43570 2/20 0.31
CA1 P00915 2/20 0.31
CA2 P00918 2/20 0.31
CA7 P43166 2/20 0.31
CA9 Q16790 2/20 0.31
CA14 Q9ULX7 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13141200 0.79 GAA (0.49) GAAKDM4EGLAMMP2MAPK1
SCHEMBL29886678 0.73 LMNA (0.43) GAAKDM4EGLAMMP2DUT
SCHEMBL28585689 0.73 RAB9A (0.43) KDM4EMMP2MAPK1LMNAALDH1A1
SCHEMBL28618725 0.73 GAA (0.53) GAAKDM4EGLAMMP2MAPK1
SCHEMBL8236144 0.73 GAA (0.53) GAAKDM4EGLAMMP2MAPK1
SCHEMBL28709031 0.72 DUT (0.38) BACE1DUTMAPT
SCHEMBL1313112 0.72 LOXL2 (0.51) GAAKDM4EMAPK1LMNAALDH1A1
SCHEMBL7367241 0.72 GAA (0.51) GAAKDM4EGLAMMP2MAPK1
SCHEMBL31132665 0.70 KDM4E (0.48) KDM4ERAB9ACA12CA1CA2
SCHEMBL28618722 0.70 KDM4E (0.50) GAAKDM4EGLAMMP2MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2534155-B1 COMPOUNDS FOR TREATING RESPIRATORY SYNCYTIAL VIRUS INFECTIONS BIOTA SCIENT MANAGEMENT PTY LTD (AU) 2018-04-11 EP disclosed
US-9540387-B2 Substituted imidazo[1,2-d]pyrrolo[1,2-d]pyrazines for treating respiratory syncytial virus infections BIOTA SCIENTIFIC MANAGEMENT PTY LTD. (AU) 2017-01-10 US disclosed
US-20160046642-A1 Compounds for Treating Respiratory Syncytial Virus Infections BIOTA SCIENT MANAGEMENT (AU) 2016-02-18 US disclosed
US-9163029-B2 Substituted imidazo[1,2-a]pyrrolo[1,2-d]pyrazines for treating respiratory syncytial virus infections BIOTA SCIENTIFIC MANAGEMENT PTY LTD. (AU) 2015-10-20 US disclosed
US-20140051697-A1 COMPOUNDS FOR TREATING RESPIRATORY SYNCYTIAL VIRUS INFECTIONS BIOTA SCIENTIFIC MANAGEMENT PTY LTD. (AU) 2014-02-20 US disclosed
US-8604034-B2 Substituted imidazo[1,2-α]pyrrolo[1,2-d]pyrazines for treating respiratory syncytial virus (RSV) infections BIOTA SCIENTIFIC MANAGEMENT PTY LTD. (AU) 2013-12-10 US disclosed
US-20110207728-A1 COMPOUNDS FOR TREATING RESPIRATORY SYNCYTIAL VIRUS INFECTIONS BIOTA SCIENTIFIC MANAGEMENT PTY LTD. (AU) 2011-08-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110207728-A1 COMPOUNDS FOR TREATING RESPIRATORY SYNCYTIAL VIRUS INFECTIONS FURIN, SQOR, SUCNR1 GAA 491/4885KDM4E 4061/4885GLA 989/4885
US-20160046642-A1 Compounds for Treating Respiratory Syncytial Virus Infections FURIN, SQOR, SUCNR1 GAA 491/4885KDM4E 4061/4885GLA 989/4885
US-20140051697-A1 COMPOUNDS FOR TREATING RESPIRATORY SYNCYTIAL VIRUS INFECTIONS FURIN, SQOR, SUCNR1 GAA 491/4885KDM4E 4061/4885GLA 989/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.