SCHEMBL2344764

SCHEMBL2344764

CCc1noc(N(C(=O)O)c2ccccc2)c1C

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.40
RAB9A P51151 4/20 0.40
LMNA P02545 1/20 0.39
TP53 P04637 1/20 0.39
MAPT P10636 1/20 0.39
TSHR P16473 3/20 0.39
NPSR1 Q6W5P4 2/20 0.38
POLB P06746 3/20 0.37
ALDH1A1 P00352 2/20 0.37
HTT P42858 1/20 0.37
KMT2A Q03164 1/20 0.37
GLA P06280 1/20 0.37
SLC26A6 Q9BXS9 2/20 0.36
L3MBTL1 Q9Y468 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2423771 0.90 NPC1 (0.38) NPC1RAB9ALMNATP53MAPT
SCHEMBL1034720 0.83 POLB (0.44) NPC1RAB9AMAPTTSHRNPSR1
SCHEMBL1081972 0.71 NPSR1 (0.41) NPC1RAB9ALMNAMAPTTSHR
SCHEMBL19778 0.67 NPSR1 (0.70) NPC1RAB9AMAPTTSHRNPSR1
SCHEMBL5590843 0.66 NPSR1 (0.47) NPC1RAB9ALMNATP53TSHR
Methylamine SCHEMBL10655180 0.65 NPSR1 (0.61) NPC1RAB9AMAPTTSHRNPSR1
SCHEMBL28335619 0.65 NPSR1 (0.50) NPC1RAB9ATSHRNPSR1POLB
SCHEMBL8705481 0.65 POLB (0.38) NPC1RAB9ATSHRNPSR1POLB
SCHEMBL8795221 0.65 EDNRB (0.42) NPC1RAB9ATP53TSHRNPSR1
SCHEMBL1037465 0.65 NPSR1 (0.41) NPC1RAB9ATSHRNPSR1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2367830-A1 1-OXA-8-AZASPIRO [4, 5] DECANE- 8 -CARBOXAMIDE COMPOUNDS AS FAAH INHIBITORS Pfizer Inc. (US) 2011-09-28 EP disclosed
US-20110230493-A1 1-OXA-8-Azaspiro [4,5] Decabe-8-Carboxamide Compounds as FAAH Inhibitors PFIZER INC. 2011-09-22 US disclosed
EP-2358704-A1 7-azaspiro [3.5]nonane-7-carboxamide compounds as modulators of fatty acid amide hydrolase Pfizer Inc. (US) 2011-08-24 EP disclosed
US-20100113465-A1 7-AZASPIRO[3.5]NONANE-7-CARBOXAMIDE COMPOUNDS PFIZER INC. 2010-05-06 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100113465-A1 7-AZASPIRO[3.5]NONANE-7-CARBOXAMIDE COMPOUNDS FAAH, FAAH2, APEH NPC1 2674/4885RAB9A 1178/4885LMNA 2680/4885
US-20110230493-A1 1-OXA-8-Azaspiro [4,5] Decabe-8-Carboxamide Compounds as FAAH Inhibitors FAAH, FAAH2, FFAR1 NPC1 2457/4885RAB9A 1697/4885LMNA 3357/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.