Sulfisoxazole

Sulfisoxazole

SCHEMBL23466

Cc1noc(NS(=O)(=O)c2ccc(N)cc2)c1C.OCCNCCO

nearest known ligand 0.79

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

folP

The experimentally established mechanism targets of Sulfisoxazole. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
EDNRA P25101 12/20 0.79
EDNRB P24530 9/20 0.79
MEN1 O00255 1/20 0.79
CYP2C9 P11712 1/20 0.79
TSHR P16473 1/20 0.79
CYP2C19 P33261 1/20 0.79
ADRA1A P35348 1/20 0.79
KMT2A Q03164 1/20 0.79

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Sulfisoxazole SCHEMBL887764 1.00 EDNRA (0.79) EDNRAEDNRBMEN1CYP2C9TSHR
Sulfisoxazole SCHEMBL3221114 0.90 EDNRA (0.82) EDNRAEDNRBMEN1CYP2C9TSHR
Sulfisoxazole SCHEMBL23467 0.89 EDNRA (1.00) EDNRAEDNRBMEN1CYP2C9TSHR
Sulfisoxazole SCHEMBL788644 0.89 EDNRA (1.00) EDNRAEDNRBMEN1CYP2C9TSHR
Sulfisoxazole SCHEMBL5917298 0.87 EDNRA (0.97) EDNRAEDNRBMEN1CYP2C9TSHR
Sulfisoxazole SCHEMBL2200933 0.87 EDNRA (0.97) EDNRAEDNRBMEN1CYP2C9TSHR
Sulfisoxazole SCHEMBL5959142 0.85 EDNRA (0.92) EDNRAEDNRBMEN1CYP2C9TSHR
Sulfisoxazole SCHEMBL16097888 0.84 EDNRA (0.89) EDNRAEDNRBMEN1CYP2C9TSHR
Sulfisoxazole SCHEMBL20770061 0.82 EDNRA (0.81) EDNRAEDNRBMEN1CYP2C9TSHR
Sulfisoxazole SCHEMBL28264710 0.82 EDNRA (0.81) EDNRAEDNRBMEN1CYP2C9TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 817 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11344506-B2 Rapidly disintegrating oral dissolvable film CUREX PHARMACEUTICAL MEXICO S.A.P.I. DE C.V. (MX) 2022-05-31 US claimed
US-20170002329-A1 GENERATING CARDIAC PROGENITOR CELLS FROM PLURIPOTENT STEM CELLS USING ISOXAZOLE OR ISOXAZOLE LIKE COMPOUNDS IPS HEART 2017-01-05 US claimed
US-20160151453-A1 METHODS AND PHARMACEUTICAL COMPOSITIONS FOR THE TREATMENT OF BACTERIAL INFECTIONS INSERM (INSTITUT NATIONAL DE LA SANTE ET DE LA RECHERCHE MEDICALE) (FR) 2016-06-02 US claimed
EP-3024476-A1 METHODS AND PHARMACEUTICAL COMPOSITIONS FOR THE TREATMENT OF BACTERIAL INFECTIONS INSERM (Institut National de la Santé et de la Recherche Médicale) (FR) 2016-06-01 EP claimed
WO-2015011254-A1 METHODS AND PHARMACEUTICAL COMPOSITIONS FOR THE TREATMENT OF BACTERIAL INFECTIONS INSERM (Institut National de la Santé et de la Recherche Médicale) (FR) 2015-01-29 WO claimed
US-20100016333-A1 Once-a-day (RNA-Polymerase Inhibiting or phenazine) - dihydropteroate synthase inhibiting - dihydrofolate reductase inhibiting antibiotic pharmaceutical product, formulation thereof, and use thereof in treating infection caused by Methicillin-Resistant Staphylococcus aureus SHIONOGI INC. 2010-01-21 US claimed
WO-2008021089-A2 ONCE-A-DAY (RNA-POLYMERASE INHIBITING OR PHENAZINE)-DIHYDROPTEROATE SYNTHASE INHIBITING-DIHYDROFOLATE REDUCTASE INHIBITING ANTIBIOTIC PHARMACEUTICAL PRODUCT, FORMULATION THEREOF, AND USE THEREOF IN TREATING INFECTION CAUSED BY METHICILLIN-RESISTANT STAPHYLOCOCCUS AUREUS MIDDLEBROOK PHARMACEUTICALS, INC. (US) 2008-02-21 WO claimed
EP-1578434-A2 METHODS AND COMPOSITIONS RELATING TO ISOLEUCINE BOROPROLINE COMPOUNDS Point Therapeutics, Inc. (US) 2005-09-28 EP claimed
US-20040131628-A1 Nucleic acids for the treatment of disorders associated with microorganisms BRATZLER ROBERT L (US) 2004-07-08 US claimed
US-20040077601-A1 Methods and compositions relating to isoleucine boroproline compounds POINT THERAPEUTICS, INC. 2004-04-22 US claimed
WO-2004004658-A2 METHODS AND COMPOSITIONS RELATING TO ISOLEUCINE BOROPROLINE COMPOUNDS POINT THERAPEUTICS, INC. (US) 2004-01-15 WO claimed
WO-2002005850-A2 ENHANCEMENT OF THE ACTION OF ANTI-INFECTIVE AGENTS PITMY INTERNATIONAL N.V. (AN) 2002-01-24 WO claimed
US-5357636-A Flexible protective medical gloves and methods for their use DRESDNER JR KARL P (US) 1994-10-25 US claimed
US-5288503-A WATER-PERMEABLE DIFFUSION BARRIER OF POLYVINYL ALCOHOL SRCHEM INCORPORATED (US) 1994-02-22 US claimed
US-5260066-A Cryogel bandage containing therapeutic agent SRCHEM INCORPORATED (US) 1993-11-09 US claimed
WO-2026107208-A1 COMPOSITIONS AND METHODS FOR TREATING MICROBIAL INFECTIONS THE METHODIST HOSPITAL (US) 2026-05-21 WO disclosed
US-20260124192-A1 COMPOUNDS, COMPOSITIONS, AND METHODS OF TREATING RNA VIRAL INFECTIONS MODEL MEDICINES INC (US) 2026-05-07 US disclosed
US-4853224-A INTRODUCING DRUG-CONTAINING POLYMERIC MICROCAPSULES INTO INTERIORS OF EYE; SUSTAINED RELEASE VISIONEX (US) 1989-08-01 US disclosed
EP-0212875-A2 Medicinal composition and method of making same Tucker, William Gough (US) 1987-03-04 EP disclosed
US-4344431-A DISPERSION OF CRYSTALLINE POLYETHYLENE AND ANTAGONIST; INSERTION INTO THE BODY-TIME-RELEASE AGENTS UNIVERSITY OF DELAWARE (US) 1982-08-17 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170002329-A1 GENERATING CARDIAC PROGENITOR CELLS FROM PLURIPOTENT STEM CELLS USING ISOXAZOLE OR ISOXAZOLE LIKE COMPOUNDS MYLK2, TNNI3, MYH2 EDNRA 3628/4885EDNRB 3227/4885MEN1 4864/4885
US-20260124192-A1 COMPOUNDS, COMPOSITIONS, AND METHODS OF TREATING RNA VIRAL INFECTIONS SARS1, NSUN2, NSUN3 EDNRA 3440/4885EDNRB 4034/4885MEN1 4294/4885
US-20040077601-A1 Methods and compositions relating to isoleucine boroproline compounds BCAT1, BCAT2, APOB EDNRA 319/4885EDNRB 110/4885MEN1 1014/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.