SCHEMBL2352302

SCHEMBL2352302

CC1(C)c2ccccc2-c2ccc(C#N)cc21

nearest known ligand 0.58

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PDK2 Q15119 3/20 0.58
PGR P06401 5/20 0.49
ALK Q9UM73 9/20 0.39
ABCC9 O60706 1/20 0.36
ABCC8 Q09428 1/20 0.36
KCNJ11 Q14654 1/20 0.36
KCNJ8 Q15842 1/20 0.36
TSHR P16473 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31295747 1.00 PDK2 (0.58) PDK2PGRALKABCC9ABCC8
SCHEMBL18914750 0.83 PGR (0.53) PDK2PGRALK
SCHEMBL13930414 0.83 PGR (0.45) PDK2PGRTSHR
SCHEMBL15158548 0.83 PGR (0.45) PDK2PGR
SCHEMBL18907195 0.82 ALDH1A1 (0.47) PDK2ALK
SCHEMBL19588872 0.82 PDK2 (0.45) PDK2PGRALK
SCHEMBL13367369 0.82 PDK2 (0.48) PDK2PGRALKTSHR
SCHEMBL10039372 0.81 PDK2 (0.61) PDK2PGRTSHR
SCHEMBL1116174 0.81 PDK2 (0.61) PDK2PGRTSHR
SCHEMBL31061764 0.81 PDK2 (0.61) PDK2PGRTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 23 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2024121084-A1 PREPARATION OF NITRILES MERCK PATENT GMBH (DE) 2024-06-13 WO disclosed
WO-2024121084-A1 PREPARATION OF NITRILES MERCK PATENT GMBH (DE) 2024-06-13 WO disclosed
US-20230126850-A1 HETEROCYCLIC SPIRO COMPOUNDS MERCK PATENT GMBH (DE) 2023-04-27 US disclosed
US-11545634-B2 Heterocyclic spiro compounds MERCK PATENT GMBH (DE) 2023-01-03 US disclosed
US-11005050-B2 Metal complexes MERCK PATENT GMBH (DE) 2021-05-11 US disclosed
EP-3708634-A1 HETEROCYCLIC SPIRO COMPOUNDS Merck Patent GmbH (DE) 2020-09-16 EP disclosed
US-10777750-B2 Heterocyclic spiro compounds BASF SE (DE) 2020-09-15 US disclosed
US-20200266364-A1 HETEROCYCLIC SPIRO COMPOUNDS MERCK PATENT GMBH (DE) 2020-08-20 US disclosed
EP-3083880-B1 HETEROCYCLIC SPIRO COMPOUNDS MERCK PATENT GMBH (DE) 2020-04-01 EP disclosed
US-20190051841-A1 HETEROCYCLIC COMPOUND AND ORGANIC LIGHT-EMITTING DEVICE INCLUDING THE SAME SAMSUNG DISPLAY CO., LTD. (KR) 2019-02-14 US disclosed
US-20160308147-A1 HETEROCYCLIC SPIRO COMPOUNDS MERCK PATENT GMBH (DE) 2016-10-20 US disclosed
US-20160260907-A1 ORGANIC ELECTROLUMINESCENT MATERIAL AND ORGANIC ELECTROLUMINESCENT DEVICE BEIJING AGLAIA TECHNOLOGY DEVELOPMENT CO., LTD. (CN) 2016-09-08 US disclosed
US-20160260907-A1 ORGANIC ELECTROLUMINESCENT MATERIAL AND ORGANIC ELECTROLUMINESCENT DEVICE BEIJING AGLAIA TECHNOLOGY DEVELOPMENT CO., LTD. (CN) 2016-09-08 US disclosed
WO-2015104045-A1 METAL COMPLEXES MERCK PATENT GMBH (DE) 2015-07-16 WO disclosed
WO-2015090504-A2 HETEROCYCLIC SPIRO COMPOUNDS MERCK PATENT GMBH (DE) 2015-06-25 WO disclosed
US-8008507-B2 Fluorescent diketopyrrolopyrroles BASF SE Ludwigshafen (DE) 2011-08-30 US disclosed
EP-1817392-B1 FLUORESCENT DIKETOPYRROLOPYRROLES CIBA HOLDING INC (CH) 2009-01-07 EP disclosed
US-20080217581-A1 Inks, colorants, pigmented plastics for coatings, non-impact-printing material, color filters, cosmetics, polymeric ink particles, toners, fluorescent tracers; high in the efficiency of electrical energy utilisation and high in luminance CIBA CORPORATION 2008-09-11 US disclosed
EP-1817392-A1 FLUORESCENT DIKETOPYRROLOPYRROLES Ciba Specialty Chemicals Holding Inc. (CH) 2007-08-15 EP disclosed
WO-2006061343-A1 FLUORESCENT DIKETOPYRROLOPYRROLES CIBA SPECIALTY CHEMICALS HOLDING INC. (CH) 2006-06-15 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (9 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20190051841-A1 HETEROCYCLIC COMPOUND AND ORGANIC LIGHT-EMITTING DEVICE INCLUDING THE SAME AOC2, CYP1A1, CRY1 PDK2 665/4885PGR 1356/4885ALK 1576/4885
US-20160308147-A1 HETEROCYCLIC SPIRO COMPOUNDS NES, KCNC1, HCN4 PDK2 264/4885PGR 1584/4885ALK 3038/4885
US-20160260907-A1 ORGANIC ELECTROLUMINESCENT MATERIAL AND ORGANIC ELECTROLUMINESCENT DEVICE APRT, TTR, ACE PDK2 1570/4885PGR 497/4885ALK 276/4885
US-11545634-B2 Heterocyclic spiro compounds NES, KCNC1, HCN4 PDK2 264/4885PGR 1584/4885ALK 3038/4885
US-20080217581-A1 Inks, colorants, pigmented plastics for coatings, non-impact-printing material, color filters, cosmetics, polymeric ink particles, toners, fluorescent tracers; high in the efficiency of electrical energy utilisation and high in luminance TYR, MC1R, IK PDK2 31/4885PGR 397/4885ALK 191/4885
US-20200266364-A1 HETEROCYCLIC SPIRO COMPOUNDS NES, KCNC1, HCN4 PDK2 264/4885PGR 1584/4885ALK 3038/4885
US-11005050-B2 Metal complexes SOD1, AP1M1, AP3M1 PDK2 2330/4885PGR 3351/4885ALK 4314/4885
US-20230126850-A1 HETEROCYCLIC SPIRO COMPOUNDS NES, KCNC1, HCN4 PDK2 264/4885PGR 1584/4885ALK 3038/4885
US-10777750-B2 Heterocyclic spiro compounds NES, KCNC1, HCN4 PDK2 264/4885PGR 1584/4885ALK 3038/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.