SCHEMBL23536190

SCHEMBL23536190

CC(=O)Nc1c(C2=CCN(c3ccc(Cl)cc3F)CC2)c(C)nn1C

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PHGDH O43175 1/20 0.39
TRPV1 Q8NER1 1/20 0.39
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
SIGMAR1 Q99720 1/20 0.35
NPC1 O15118 1/20 0.34
HTT P42858 2/20 0.34
DRD4 P21917 1/20 0.34
GRM2 Q14416 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
PROKR1 Q8TCW9 1/20 0.34
RXFP1 Q9HBX9 1/20 0.34
MAPT P10636 3/20 0.33
IDO1 P14902 1/20 0.33
TDO2 P48775 1/20 0.33
C5AR1 P21730 1/20 0.33
GRM5 P41594 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29932049 1.00 PHGDH (0.39) PHGDHTRPV1MEN1KMT2ASIGMAR1
SCHEMBL29932026 0.81 SIGMAR1 (0.36) PHGDHTRPV1SIGMAR1DRD4GRM2
SCHEMBL29931958 0.79 DRD4 (0.38) PHGDHTRPV1SIGMAR1DRD4GRM2
SCHEMBL23536237 0.79 DRD4 (0.38) PHGDHTRPV1SIGMAR1DRD4GRM2
SCHEMBL29932124 0.79 PHGDH (0.42) PHGDHMEN1KMT2AHTTPROKR1
SCHEMBL23536493 0.79 PHGDH (0.42) PHGDHMEN1KMT2AHTTPROKR1
SCHEMBL23536369 0.77 ALDH1A1 (0.38) PHGDHMEN1KMT2ADRD4GRM2
SCHEMBL29932109 0.73 MAPT (0.37) MEN1KMT2AHTTCYP3A4CYP2C9
SCHEMBL29931836 0.71 GAA (0.34) KMT2AHTTDRD4GRM2PROKR1
SCHEMBL23536396 0.64 ALDH1A1 (0.39) TRPV1SIGMAR1HTTDRD4GRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115087440-A TRPML modulators 卡斯玛治疗公司 2022-09-20 CN disclosed
WO-2021127337-A1 TRPML MODULATORS CASMA THERAPEUTICS, INC. (US) 2021-06-24 WO disclosed