SCHEMBL23536408

SCHEMBL23536408

CC(=O)c1cccc(F)c1N1CCC2(CC1)COC(C)(C)C2

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPK8 P45983 1/20 0.34
MAPK10 P53779 1/20 0.34
USP2 O75604 3/20 0.34
KMT2A Q03164 2/20 0.33
GPR119 Q8TDV5 2/20 0.33
PGR P06401 1/20 0.33
HPGD P15428 2/20 0.33
AVPR1A P37288 2/20 0.32
MAPK1 P28482 3/20 0.32
CYP1A2 P05177 2/20 0.32
HSD17B10 Q99714 2/20 0.32
SMN1; SMN2 Q16637 2/20 0.32
SPR P35270 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C19 P33261 2/20 0.32
ALDH1A1 P00352 2/20 0.32
MEN1 O00255 1/20 0.32
CYP3A4 P08684 1/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29931913 1.00 MAPK8 (0.34) MAPK8MAPK10USP2KMT2AGPR119
SCHEMBL23555192 0.81 MC4R (0.32) GPR119
SCHEMBL23536132 0.81
SCHEMBL23535948 0.80 ICMT (0.32) GPR119
SCHEMBL23536133 0.80 ICMT (0.31) GPR119
SCHEMBL23536144 0.79 GPR119 (0.31) GPR119
SCHEMBL29932063 0.79 KMT2A (0.39) KMT2AHPGDSMN1; SMN2ALDH1A1NPC1
SCHEMBL23536595 0.76 GPR119 (0.38) KMT2AGPR119MEN1
SCHEMBL29948426 0.76 GPR119 (0.38) KMT2AGPR119MEN1
SCHEMBL18412770 0.74 ALDH1A1 (0.55) HPGDHSD17B10SMN1; SMN2ALDH1A1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230104936-A1 TRPML MODULATORS CASMA THERAPEUTICS, INC. 2023-04-06 US disclosed
WO-2021127337-A1 TRPML MODULATORS CASMA THERAPEUTICS, INC. (US) 2021-06-24 WO disclosed
WO-2021127337-A1 TRPML MODULATORS CASMA THERAPEUTICS, INC. (US) 2021-06-24 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230104936-A1 TRPML MODULATORS TRPM2, TRPM4, TRPM5 MAPK8 2158/4885MAPK10 1014/4885USP2 4313/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.