SCHEMBL2355313

SCHEMBL2355313

COCC(=O)N(C(=O)C1CCCN1)c1ccc(Oc2ccc(F)cc2)cc1

nearest known ligand 0.45

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 2/20 0.45
HTR2B P41595 1/20 0.45
PFKFB3 Q16875 4/20 0.42
PFKFB1 P16118 3/20 0.42
PFKFB2 O60825 2/20 0.42
LTA4H P09960 1/20 0.40
MLNR O43193 3/20 0.37
SCN4A P35499 1/20 0.37
KCNH2 Q12809 1/20 0.36
DPP4 P27487 3/20 0.35
KMT2A Q03164 1/20 0.35
TACR1 P25103 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2170198 0.90 HTR2C (0.41) HTR2CHTR2BPFKFB3PFKFB1PFKFB2
SCHEMBL2170165 0.83 HTR2C (0.46) HTR2CHTR2BPFKFB3PFKFB1PFKFB2
SCHEMBL2353722 0.81 HTR2C (0.41) HTR2CHTR2BPFKFB3PFKFB1PFKFB2
SCHEMBL2171149 0.80 HTR2C (0.41) HTR2CHTR2BPFKFB3PFKFB1PFKFB2
SCHEMBL2356689 0.80 HRH3 (0.44) HTR2CHTR2BPFKFB3PFKFB1PFKFB2
SCHEMBL2364515 0.78 HTR2C (0.39) HTR2CHTR2BPFKFB3PFKFB1PFKFB2
SCHEMBL2170010 0.77 HTR2C (0.39) HTR2CHTR2BPFKFB3PFKFB1PFKFB2
SCHEMBL2352725 0.76 HTR2C (0.41) HTR2CHTR2BPFKFB3PFKFB1PFKFB2
SCHEMBL29517131 0.72 SCN4A (0.58) PFKFB3PFKFB1PFKFB2MLNRSCN4A
SCHEMBL26364702 0.72 SCN4A (0.58) PFKFB3PFKFB1PFKFB2MLNRSCN4A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2349252-A2 SYNERGISTIC COMBINATION OF SPHINGOSINE-1-PHOSPHATE RECEPTOR ANTAGONISTS AND ANTIMICROTUBULE AGENTS Exelixis, Inc. (US) 2011-08-03 EP disclosed