SCHEMBL2170198

SCHEMBL2170198

COCCC(=O)N(C(=O)C1CCCN1)c1ccc(Oc2ccc(F)cc2)cc1

nearest known ligand 0.41

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 2/20 0.41
HTR2B P41595 1/20 0.41
PFKFB2 O60825 1/20 0.41
PFKFB1 P16118 1/20 0.41
PFKFB3 Q16875 1/20 0.41
LTA4H P09960 2/20 0.38
MLNR O43193 4/20 0.37
SCN4A P35499 1/20 0.36
DPP4 P27487 4/20 0.36
KCNH2 Q12809 1/20 0.35
ALDH1A1 P00352 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2355313 0.90 HTR2C (0.45) HTR2CHTR2BPFKFB2PFKFB1PFKFB3
SCHEMBL2170165 0.84 HTR2C (0.46) HTR2CHTR2BPFKFB2PFKFB1PFKFB3
SCHEMBL2353722 0.83 HTR2C (0.41) HTR2CHTR2BPFKFB2PFKFB1PFKFB3
SCHEMBL2364515 0.80 HTR2C (0.39) HTR2CHTR2BPFKFB2PFKFB1PFKFB3
SCHEMBL2171149 0.79 HTR2C (0.41) HTR2CHTR2BPFKFB2PFKFB1PFKFB3
SCHEMBL2356689 0.79 HRH3 (0.44) HTR2CHTR2BPFKFB2PFKFB1PFKFB3
SCHEMBL2353030 0.78 OPRM1 (0.37)
SCHEMBL2170010 0.76 HTR2C (0.39) HTR2CHTR2BPFKFB2PFKFB1PFKFB3
SCHEMBL2352725 0.75 HTR2C (0.41) HTR2CHTR2BPFKFB2PFKFB1PFKFB3
SCHEMBL2354130 0.71 OPRM1 (0.38) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2346821-A1 SPHINGOSINE-1-PHOSPHATE RECEPTOR ANTAGONISTS Exelixis, Inc. (US) 2011-07-27 EP disclosed