SCHEMBL2353722

SCHEMBL2353722

O=C(CCC(=O)N(C(=O)C1CCCN1)c1ccc(Oc2ccc(F)cc2)cc1)c1ccccc1

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 2/20 0.41
HTR2B P41595 2/20 0.41
PFKFB2 O60825 1/20 0.38
PFKFB1 P16118 1/20 0.38
PFKFB3 Q16875 1/20 0.38
KMT2A Q03164 2/20 0.36
LTA4H P09960 1/20 0.36
MMP1 P03956 1/20 0.36
MLNR O43193 3/20 0.35
SCN4A P35499 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
DPP4 P27487 2/20 0.34
DPP8 Q6V1X1 1/20 0.34
MEN1 O00255 1/20 0.33
ALDH1A1 P00352 1/20 0.33
POLB P06746 1/20 0.33
ANPEP P15144 1/20 0.33
DRD2 P14416 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2364515 0.85 HTR2C (0.39) HTR2CHTR2BPFKFB2PFKFB1PFKFB3
SCHEMBL2170165 0.85 HTR2C (0.46) HTR2CHTR2BPFKFB2PFKFB1PFKFB3
SCHEMBL2170198 0.83 HTR2C (0.41) HTR2CHTR2BPFKFB2PFKFB1PFKFB3
SCHEMBL2355313 0.81 HTR2C (0.45) HTR2CHTR2BPFKFB2PFKFB1PFKFB3
SCHEMBL2352725 0.78 HTR2C (0.41) HTR2CHTR2BPFKFB2PFKFB1PFKFB3
SCHEMBL2171149 0.78 HTR2C (0.41) HTR2CHTR2BPFKFB2PFKFB1PFKFB3
SCHEMBL2356689 0.76 HRH3 (0.44) HTR2CHTR2BPFKFB2PFKFB1PFKFB3
SCHEMBL2170010 0.73 HTR2C (0.39) HTR2CHTR2BPFKFB2PFKFB1PFKFB3
SCHEMBL2353030 0.69 OPRM1 (0.37) KMT2AMEN1POLB
SCHEMBL11158703 0.68 KMT2A (0.43) KMT2AL3MBTL1MEN1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2349252-A2 SYNERGISTIC COMBINATION OF SPHINGOSINE-1-PHOSPHATE RECEPTOR ANTAGONISTS AND ANTIMICROTUBULE AGENTS Exelixis, Inc. (US) 2011-08-03 EP disclosed