SCHEMBL2364515

SCHEMBL2364515

O=C(CCC(=O)N(C(=O)C1CCCN1)c1ccc(Oc2ccc(F)cc2)cc1)c1cccs1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 1/20 0.39
HTR2B P41595 1/20 0.39
ALDH1A1 P00352 3/20 0.38
LMNA P02545 2/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
NPC1 O15118 1/20 0.38
POLB P06746 1/20 0.38
RAB9A P51151 1/20 0.38
CTNNB1 P35222 2/20 0.36
WNT3A P56704 2/20 0.36
PFKFB2 O60825 1/20 0.36
PFKFB1 P16118 1/20 0.36
PFKFB3 Q16875 1/20 0.36
CYP1A2 P05177 1/20 0.34
CYP2D6 P10635 1/20 0.34
LTA4H P09960 1/20 0.34
MAPT P10636 1/20 0.34
MAPK1 P28482 1/20 0.34
KCNA5 P22460 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2353722 0.85 HTR2C (0.41) HTR2CHTR2BALDH1A1MEN1KMT2A
SCHEMBL2171149 0.84 HTR2C (0.41) HTR2CHTR2BALDH1A1LMNAMEN1
SCHEMBL2170198 0.80 HTR2C (0.41) HTR2CHTR2BALDH1A1PFKFB2PFKFB1
SCHEMBL2170165 0.78 HTR2C (0.46) HTR2CHTR2BMEN1KMT2APFKFB2
SCHEMBL2355313 0.78 HTR2C (0.45) HTR2CHTR2BKMT2APFKFB2PFKFB1
SCHEMBL2356689 0.73 HRH3 (0.44) HTR2CHTR2BALDH1A1LMNAKMT2A
SCHEMBL2352725 0.72 HTR2C (0.41) HTR2CHTR2BPFKFB2PFKFB1PFKFB3
SCHEMBL2170010 0.71 HTR2C (0.39) HTR2CHTR2BPFKFB2PFKFB1PFKFB3
SCHEMBL11231004 0.70 ALDH1A1 (0.50) ALDH1A1LMNAMEN1KMT2ANPC1
SCHEMBL4164203 0.65 TSHR (0.46) ALDH1A1LMNAMEN1KMT2ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2349252-A2 SYNERGISTIC COMBINATION OF SPHINGOSINE-1-PHOSPHATE RECEPTOR ANTAGONISTS AND ANTIMICROTUBULE AGENTS Exelixis, Inc. (US) 2011-08-03 EP disclosed
WO-2010045601-A2 SYNERGISTIC EFFECTS BETWEEN SPHINGOSINE-1-PHOSPHATE RECEPTOR ANTAGONISTS AND ANTIMICROTUBULE AGENTS EXELIXIS, INC. (US) 2010-04-22 WO disclosed