SCHEMBL2356689

SCHEMBL2356689

O=C(CN1CCOCC1)N(C(=O)C1CCCN1)c1ccc(Oc2ccc(F)cc2)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 2/20 0.44
ALDH1A1 P00352 3/20 0.40
HPGD P15428 2/20 0.40
ALOX15 P16050 1/20 0.40
MLNR O43193 4/20 0.40
HTR2C P28335 1/20 0.39
HTR2B P41595 1/20 0.39
PFKFB2 O60825 1/20 0.39
PFKFB1 P16118 1/20 0.39
PFKFB3 Q16875 1/20 0.39
ATM Q13315 1/20 0.39
KMT2A Q03164 1/20 0.37
LMNA P02545 1/20 0.37
TP53 P04637 1/20 0.37
FKBP1A P62942 1/20 0.36
PIK3CD O00329 1/20 0.36
PIK3CA P42336 1/20 0.36
PIK3CB P42338 1/20 0.36
PIK3CG P48736 1/20 0.36
LTA4H P09960 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2355313 0.80 HTR2C (0.45) MLNRHTR2CHTR2BPFKFB2PFKFB1
SCHEMBL2170010 0.79 HTR2C (0.39) MLNRHTR2CHTR2BPFKFB2PFKFB1
SCHEMBL2170165 0.79 HTR2C (0.46) MLNRHTR2CHTR2BPFKFB2PFKFB1
SCHEMBL2170198 0.79 HTR2C (0.41) ALDH1A1MLNRHTR2CHTR2BPFKFB2
SCHEMBL2171149 0.77 HTR2C (0.41) ALDH1A1HPGDHTR2CHTR2BPFKFB2
SCHEMBL2353722 0.76 HTR2C (0.41) ALDH1A1MLNRHTR2CHTR2BPFKFB2
SCHEMBL2364515 0.73 HTR2C (0.39) ALDH1A1HTR2CHTR2BPFKFB2PFKFB1
SCHEMBL2352725 0.72 HTR2C (0.41) HTR2CHTR2BPFKFB2PFKFB1PFKFB3
SCHEMBL2350633 0.70 OPRM1 (0.39) HRH3ALDH1A1KMT2ALMNASCN9A
SCHEMBL23373319 0.67 PFKFB3 (0.53) HRH3ALDH1A1HPGDALOX15PFKFB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2349252-A2 SYNERGISTIC COMBINATION OF SPHINGOSINE-1-PHOSPHATE RECEPTOR ANTAGONISTS AND ANTIMICROTUBULE AGENTS Exelixis, Inc. (US) 2011-08-03 EP disclosed