SCHEMBL2171155

SCHEMBL2171155

NC(=O)C1CCCN1C(=O)C(c1ccc(Oc2ccc(F)cc2)cc1)c1cccs1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 5/20 0.52
FPR2 P25090 2/20 0.42
DPP4 P27487 1/20 0.39
RAB9A P51151 1/20 0.39
MAOA P21397 1/20 0.38
MAOB P27338 1/20 0.38
HTR1A P08908 1/20 0.38
HTR7 P34969 1/20 0.38
FKBP4 Q02790 1/20 0.38
FKBP5 Q13451 1/20 0.38
CHRM2 P08172 1/20 0.36
CHRM1 P11229 1/20 0.36
CHRM3 P20309 1/20 0.36
SCN3A Q9NY46 1/20 0.36
PDE4A P27815 1/20 0.36
PDE4B Q07343 1/20 0.36
PDE4C Q08493 1/20 0.36
PDE4D Q08499 1/20 0.36
KCNH2 Q12809 1/20 0.36
APOL1 O14791 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2170169 0.86 SCN9A (0.54) SCN9AFPR2DPP4RAB9A
SCHEMBL2355316 0.77 SCN9A (0.52) SCN9AFPR2DPP4RAB9AHTR1A
SCHEMBL13570422 0.76 CES2 (0.41) DPP4RAB9ACHRM2CHRM1CHRM3
SCHEMBL2356691 0.74 SCN9A (0.48) SCN9AFPR2DPP4RAB9AHTR1A
SCHEMBL6980126 0.72 AGTR2 (0.52) DPP4
SCHEMBL2170202 0.71 SCN9A (0.49) SCN9AFPR2DPP4HTR1AHTR7
SCHEMBL2364602 0.69 HTR2C (0.45) CHRM2CHRM1CHRM3PDE4APDE4B
SCHEMBL2172455 0.69 SCN9A (0.60) SCN9AFPR2DPP4HTR1AHTR7
Hydrochloric Acid SCHEMBL2169819 0.68 SCN9A (0.59) SCN9AFPR2DPP4HTR1AHTR7
SCHEMBL2352727 0.68 SCN9A (0.53) SCN9AFPR2DPP4HTR1AHTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2346821-A1 SPHINGOSINE-1-PHOSPHATE RECEPTOR ANTAGONISTS Exelixis, Inc. (US) 2011-07-27 EP disclosed