SCHEMBL237290

SCHEMBL237290

CC(=O)c1cccc(OCc2c(C)cccc2C)c1

nearest known ligand 0.67

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
MAOB P27338 14/20 0.67
MAOA P21397 4/20 0.61
KMT2A Q03164 2/20 0.51
MEN1 O00255 1/20 0.51
SMN1; SMN2 Q16637 1/20 0.51
ABCB1 P08183 1/20 0.49
SLC22A12 Q96S37 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2086718 0.90 MAOB (0.61) MAOBMAOAKMT2AMEN1SMN1; SMN2
SCHEMBL1633991 0.88 NR4A2 (0.65) KMT2A
SCHEMBL31215373 0.88 NR4A2 (0.65) KMT2A
SCHEMBL2087954 0.85 MAOB (0.71) MAOBMAOA
SCHEMBL955309 0.85 MAOB (0.51) MAOBKMT2ASMN1; SMN2SLC22A12
SCHEMBL2089424 0.84 MAOB (0.69) MAOBMAOASMN1; SMN2
SCHEMBL1634331 0.84 TDP1 (0.52) MAOBKMT2AMEN1SMN1; SMN2
SCHEMBL235381 0.84 MAOB (0.48) MAOBMAOASMN1; SMN2SLC22A12
SCHEMBL237424 0.84 MAOB (0.48) MAOBMAOASMN1; SMN2SLC22A12
SCHEMBL1437471 0.83 MAOB (0.68) MAOBMAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 82 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2285777-B1 SYNTHESIS OF 4-[3-(2,6-DIMETHYLBENZYLOXY)PHENYL]-4-OXOBUTANOIC ACID WELLSTAT THERAPEUTICS CORP (US) 2016-09-07 EP claimed
US-8703991-B2 Synthesis of (phenylalkyloxy)phenyl-oxobutanoic acids WELLSTAT THERAPEUTICS CORPORATION (US) 2014-04-22 US claimed
US-8664433-B2 Synthesis of 4-[3-(2,6-dimethylbenzyloxy)phenyl]-4-oxobutanoic acid WELLSTAT THERAPEUTICS CORPORATION (US) 2014-03-04 US claimed
US-20120004442-A1 SYNTHESIS OF (PHENYLALKYLOXY)PHENYL-OXOBUTANOIC ACIDS WELLSTAT THERAPEUTICS CORPORATION (US) 2012-01-05 US claimed
EP-2365746-A1 SYNTHESIS OF (PHENYLALKYLOXY)PHENYL-OXOBUTANOIC ACIDS Wellstat Therapeutics Corporation (US) 2011-09-21 EP claimed
US-20110201838-A1 SYNTHESIS OF 4-[3-(2,6-DIMETHYLBENZYLOXY)PHENYL]-4-OXOBUTANOIC ACID WELLSTAT THERAPEUTICS CORPORATION (US) 2011-08-18 US claimed
WO-2010053910-A1 SYNTHESIS OF (PHENYLALKYLOXY)PHENYL-OXOBUTANOIC ACIDS WELLSTAT THERAPEUTICS CORPORATION (US) 2010-05-14 WO claimed
WO-2009137381-A1 SYNTHESIS OF 4-[3-(2,6-DIMETHYLBENZYLOXY)PHENYL]-4-OXOBUTANOIC ACID WELLSTAT THERAPEUTICS CORPORATION (US) 2009-11-12 WO claimed
EP-3517109-A1 COMPOUNDS AND METHOD FOR REDUCING URIC ACID Wellstat Therapeutics Corporation (US) 2019-07-31 EP disclosed
EP-2268141-B1 COMPOUND AND METHOD FOR REDUCING URIC ACID WELLSTAT THERAPEUTICS CORP (US) 2019-05-08 EP disclosed
EP-2285777-B1 SYNTHESIS OF 4-[3-(2,6-DIMETHYLBENZYLOXY)PHENYL]-4-OXOBUTANOIC ACID WELLSTAT THERAPEUTICS CORP (US) 2016-09-07 EP disclosed
US-9133073-B2 Compounds for the treatment of metabolic disorders WELLSTAT THERAPEUTICS CORPORATION (US) 2015-09-15 US disclosed
US-9115072-B2 Compounds and method for reducing uric acid WELLSTAT THERAPEUTICS CORPORATION (US) 2015-08-25 US disclosed
US-8829058-B2 Compounds and method for reducing uric acid WELLSTAT THERAPEUTICS CORPORATION (US) 2014-09-09 US disclosed
US-20040097585-A1 Compounds for the treatment of metabolic disorders WELLSTAT THERAPEUTICS CORPORATION 2004-05-20 US disclosed
US-20040092516-A1 Compounds for the treatment of metabolic disorders PHARMA CINQ, LLC 2004-05-13 US disclosed
US-20040092518-A1 Compounds for the treatment of metabolic disorders PHARMA CINQ, LLC 2004-05-13 US disclosed
US-20040077896-A1 Compounds for the treatment of metabolic disorders WELLSTAT THERAPEUTICS CORPORATION 2004-04-22 US disclosed
US-20030149107-A1 Compounds for the treatment of metabolic disorders PHARMA CINQ, LLC 2003-08-07 US disclosed
WO-2002100341-A2 COMPOUNDS FOR THE TREATMENT OF METABOLIC DISORDERS WELLSTAT THERAPEUTICS CORPORATION (US) 2002-12-19 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (7 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20040092516-A1 Compounds for the treatment of metabolic disorders GOT2, OAT, CPT1B MAOB 589/4885MAOA 1265/4885KMT2A 3364/4885
US-20120004442-A1 SYNTHESIS OF (PHENYLALKYLOXY)PHENYL-OXOBUTANOIC ACIDS PGD, HPD, MLYCD MAOB 684/4885MAOA 1278/4885KMT2A 2740/4885
US-20040092518-A1 Compounds for the treatment of metabolic disorders GOT2, OAT, CPT1B MAOB 589/4885MAOA 1265/4885KMT2A 3364/4885
US-20040097585-A1 Compounds for the treatment of metabolic disorders GOT2, OAT, CPT1B MAOB 589/4885MAOA 1265/4885KMT2A 3364/4885
US-20110201838-A1 SYNTHESIS OF 4-[3-(2,6-DIMETHYLBENZYLOXY)PHENYL]-4-OXOBUTANOIC ACID HPD, EIF4B, MVD MAOB 223/4885MAOA 1091/4885KMT2A 2879/4885
US-20040077896-A1 Compounds for the treatment of metabolic disorders GOT2, OAT, CPT1B MAOB 589/4885MAOA 1265/4885KMT2A 3364/4885
US-20030149107-A1 Compounds for the treatment of metabolic disorders GOT2, OAT, CPT1B MAOB 589/4885MAOA 1265/4885KMT2A 3364/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.