SCHEMBL23730754

SCHEMBL23730754

CC(C)n1c(Br)nc2[nH]c(=O)[nH]c(=O)c21

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GDA Q9Y2T3 1/20 0.40
MEN1 O00255 3/20 0.34
KMT2A Q03164 3/20 0.34
ALDH1A1 P00352 6/20 0.33
HSD17B10 Q99714 4/20 0.33
HPGD P15428 3/20 0.33
KDM4E B2RXH2 2/20 0.33
MAPT P10636 2/20 0.33
ALOX15 P16050 1/20 0.33
ALOX12 P18054 1/20 0.33
DPP4 P27487 1/20 0.33
RPS6KA3 P51812 1/20 0.31
CYP1A2 P05177 2/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
BRDT Q58F21 1/20 0.30
NOD1 Q9Y239 1/20 0.30
GAA P10253 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30
ADORA3 P0DMS8 1/20 0.30
ADORA2A P29274 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18989874 0.77 GDA (0.47) GDAALDH1A1HSD17B10KDM4EMAPT
SCHEMBL21389576 0.73 GDA (0.40) GDAMEN1KMT2AALDH1A1KDM4E
SCHEMBL27908390 0.68 NOD1 (0.37) GDAMEN1KMT2AALDH1A1KDM4E
SCHEMBL15519472 0.66 KDM4E (0.38) GDAALDH1A1HPGDKDM4EMAPT
SCHEMBL7004955 0.65 GDA (0.49) GDAALDH1A1HSD17B10KDM4EMAPT
SCHEMBL20097140 0.64 GDA (0.62) GDAMEN1KMT2AALDH1A1HSD17B10
SCHEMBL22105384 0.64 DPP4 (0.62) MEN1KMT2AALDH1A1KDM4EMAPT
SCHEMBL4037097 0.61 GDA (0.41) GDAMEN1KMT2AALDH1A1HSD17B10
SCHEMBL1833932 0.60 POLB (0.47) MEN1KMT2AALDH1A1HSD17B10HPGD
SCHEMBL517356 0.59 MAPT (0.46) GDAMEN1KMT2AALDH1A1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3397640-B1 XANTHINE DERIVATIVE INHIBITORS OF BET PROTEINS INST NAT SANTE RECH MED (FR) 2021-08-04 EP disclosed