SCHEMBL2373864

SCHEMBL2373864

O=C(O)c1c(CBr)c(-c2cccc(C(F)(F)F)c2)nc2ccc(Cl)cc12

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 9/20 0.54
CYP2C9 P11712 3/20 0.48
ALDH1A1 P00352 2/20 0.48
GAA P10253 1/20 0.48
KDM4E B2RXH2 2/20 0.45
CYP1A2 P05177 2/20 0.45
CYP2C19 P33261 2/20 0.45
HTT P42858 2/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
LMNA P02545 1/20 0.45
CYP3A4 P08684 1/20 0.45
NLRP3 Q96P20 1/20 0.45
FABP3 P05413 2/20 0.43
FABP4 P15090 2/20 0.43
FABP5 Q01469 1/20 0.43
MEN1 O00255 1/20 0.43
CYP2D6 P10635 1/20 0.43
KMT2A Q03164 1/20 0.43
PTGFR P43088 4/20 0.42
IP6K1 Q92551 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2372472 0.89 PLA2G2A (0.51) DHODHCYP2C9ALDH1A1GAAKDM4E
SCHEMBL2372767 0.88 DHODH (0.56) DHODH
SCHEMBL2372279 0.87 DHODH (0.50) DHODHLMNA
SCHEMBL2372504 0.85 DHODH (0.69) DHODHCYP2C9ALDH1A1GAAKDM4E
SCHEMBL5908732 0.84 DHODH (0.67) DHODHPTGFR
SCHEMBL2373216 0.81 LMNA (0.51) DHODHCYP2C9KDM4ECYP1A2CYP2C19
SCHEMBL2373306 0.80 DHODH (0.51) DHODHCYP2C9ALDH1A1KDM4ECYP1A2
SCHEMBL5908769 0.79 DHODH (0.57) DHODHCYP2C9CYP1A2CYP2C19LMNA
SCHEMBL2373738 0.78 TRPV4 (0.67)
SCHEMBL2373037 0.77 DHODH (0.70) DHODHCYP2C9KDM4ECYP1A2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011119693-A1 TRPV4 ANTAGONISTS GLAXOSMITHKLINE LLC (US) 2011-09-29 WO disclosed