SCHEMBL23747465

SCHEMBL23747465

CN1CCN(Cc2ccc(NC(=O)NCc3ccc(Cl)cc3)cc2F)CC1=O

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 2/20 0.48
CHRM1 P11229 1/20 0.48
MCHR1 Q99705 1/20 0.48
RAB9A P51151 3/20 0.48
POLB P06746 3/20 0.48
NPC1 O15118 1/20 0.46
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
MAPT P10636 1/20 0.44
NAMPT P43490 2/20 0.43
LSS P48449 1/20 0.43
CNR1 P21554 1/20 0.43
LMNA P02545 1/20 0.42
HPGD P15428 1/20 0.42
TSHR P16473 1/20 0.42
ERCC1 P07992 1/20 0.42
ERCC4 Q92889 1/20 0.42
EPHX2 P34913 1/20 0.41
DDB1 Q16531 1/20 0.41
CRBN Q96SW2 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26101837 0.87 CHRM1 (0.62) HTR2ACHRM1MCHR1RAB9APOLB
SCHEMBL23747349 0.83 RAB9A (0.48) HTR2ACHRM1MCHR1RAB9APOLB
SCHEMBL23747463 0.83 CHRM1 (0.45) HTR2ACHRM1MCHR1RAB9APOLB
SCHEMBL26100896 0.80 CHRM1 (0.53) HTR2ACHRM1MCHR1RAB9APOLB
SCHEMBL24024157 0.73 NOD1 (0.62) RAB9ANPC1MEN1KMT2AMAPT
SCHEMBL23747450 0.71 RAB9A (0.52) HTR2ACHRM1MCHR1RAB9APOLB
SCHEMBL26101687 0.71 RAB9A (0.57) HTR2ACHRM1MCHR1RAB9APOLB
SCHEMBL23747696 0.71 SMN1; SMN2 (0.63) HTR2ACHRM1MCHR1RAB9APOLB
SCHEMBL23747451 0.71 RAB9A (0.54) RAB9APOLBNPC1MEN1KMT2A
SCHEMBL23747697 0.71 L3MBTL1 (0.45) HTR2ACHRM1MCHR1RAB9AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230133132-A1 NAMPT MODULATORS CYTOKINETICS, INC. 2023-05-04 US disclosed
US-20230133132-A1 NAMPT MODULATORS CYTOKINETICS, INC. 2023-05-04 US disclosed
US-20230133132-A1 NAMPT MODULATORS CYTOKINETICS, INC. 2023-05-04 US disclosed
WO-2021159015-A1 NAMPT MODULATORS CYTOKINETICS, INC. (US) 2021-08-12 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230133132-A1 NAMPT MODULATORS NAMPT, MC4R, SIRT1 HTR2A 2115/4885CHRM1 1155/4885MCHR1 358/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.