SCHEMBL23770596

SCHEMBL23770596

Cc1ccc(F)cc1-c1nc(NSc2ccnc(N3CCNCC3)c2)ccc1C(F)(F)F

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRB1 P08588 1/20 0.41
CYP1A2 P05177 3/20 0.39
CYP2C9 P11712 1/20 0.39
KARS1 Q15046 3/20 0.39
CYP2C19 P33261 1/20 0.37
ABL1 P00519 1/20 0.36
RAF1 P04049 1/20 0.36
BRAF P15056 1/20 0.36
ADRB2 P07550 1/20 0.36
HTR2C P28335 2/20 0.35
ALK Q9UM73 1/20 0.34
CDK4 P11802 3/20 0.34
CCND1 P24385 3/20 0.34
CDK1 P06493 1/20 0.34
CCNB1 P14635 1/20 0.34
CCNA2 P20248 1/20 0.34
CDK2 P24941 1/20 0.34
CCNA1 P78396 1/20 0.34
NCF1 P14598 1/20 0.34
SOS1 Q07889 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23770587 0.88 ABL1 (0.39) ADRB1CYP1A2KARS1ABL1HTR2C
SCHEMBL23770583 0.86 RAF1 (0.36) ABL1RAF1BRAFSOS1
SCHEMBL23770447 0.85 SOS1 (0.34) ABL1RAF1BRAFSOS1
SCHEMBL23770770 0.84 ADRB2 (0.38) CYP1A2CYP2C9KARS1CYP2C19ABL1
SCHEMBL19951363 0.82 NMT1 (0.41) ADRB1CYP1A2CYP2C9KARS1ABL1
SCHEMBL23770773 0.82 ABL1 (0.37) ABL1
SCHEMBL23770701 0.80 ATR (0.42) RAF1BRAF
SCHEMBL23770607 0.77 JAK2 (0.35) ABL1CCNA2CDK2CCNA1
SCHEMBL23770452 0.76 PDE10A (0.34) ABL1
SCHEMBL23770466 0.75 CYP1A2 (0.37) CYP1A2CYP2C19ABL1CCNA2CDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3504194-B1 N-(PYRIDIN-2-YL)PYRIDINE-SULFONAMIDE DERIVATIVES AND THEIR USE IN THE TREATMENT OF DISEASE NOVARTIS AG (CH) 2021-08-18 EP disclosed