SCHEMBL23770652

SCHEMBL23770652

Cc1ccc(C#N)cc1-c1nc(NSc2cccc(N)n2)ccc1C(F)(F)F

nearest known ligand 0.32

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 1/20 0.32
TRPA1 O75762 1/20 0.31
CDC7 O00311 1/20 0.31
CDK2 P24941 1/20 0.31
PTGDR2 Q9Y5Y4 1/20 0.31
KDM4E B2RXH2 1/20 0.30
ALDH1A1 P00352 1/20 0.30
TDP1 Q9NUW8 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30
AR P10275 1/20 0.30
ACP1 P24666 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23770566 0.86 AGPAT2 (0.35) TRPA1
SCHEMBL23770740 0.85 HSD11B1 (0.33) HSD11B1CDC7CDK2AR
SCHEMBL23770551 0.85 PTPN1 (0.36) TRPA1ALDH1A1AR
SCHEMBL23770604 0.83 DHFR (0.32)
SCHEMBL23770684 0.83 ADRB2 (0.36) ALDH1A1
SCHEMBL23770544 0.82 S1PR1 (0.33) CDC7CDK2PTGDR2
SCHEMBL23770405 0.81 PTPN1 (0.31)
SCHEMBL23770666 0.80 KRAS (0.39) PTGDR2KDM4EALDH1A1AR
SCHEMBL29464398 0.80 HSD11B1 (0.43) HSD11B1KDM4E
SCHEMBL19968784 0.80 HSD11B1 (0.43) HSD11B1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3504194-B1 N-(PYRIDIN-2-YL)PYRIDINE-SULFONAMIDE DERIVATIVES AND THEIR USE IN THE TREATMENT OF DISEASE NOVARTIS AG (CH) 2021-08-18 EP disclosed