SCHEMBL23770769

SCHEMBL23770769

COc1ccccc1-c1nc(NSc2cccc(N)n2)ccc1Cl

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.38
ADORA2A P29274 3/20 0.38
HSP90AA1 P07900 2/20 0.38
HSP90AB1 P08238 1/20 0.38
ADORA1 P30542 2/20 0.37
HSD17B10 Q99714 1/20 0.36
HTR1A P08908 1/20 0.36
HTR1D P28221 1/20 0.36
HTR1B P28222 1/20 0.36
HTR2A P28223 1/20 0.36
HTR2C P28335 1/20 0.36
HTR1E P28566 1/20 0.36
HTR7 P34969 1/20 0.36
HTR2B P41595 1/20 0.36
HTR5A P47898 1/20 0.36
HTR6 P50406 1/20 0.36
HPGD P15428 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
GAA P10253 2/20 0.34
KDM4E B2RXH2 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23770637 0.89 PDE4B (0.38) HSP90AA1HSP90AB1AGPAT2
SCHEMBL23770590 0.86 ADORA2A (0.35) ADORA2AHSP90AA1GAALMNADPP4
SCHEMBL23770591 0.86 SCN10A (0.38)
SCHEMBL23770409 0.86 BACE1 (0.35) ALDH1A1HSP90AA1HSP90AB1GAAKDM4E
SCHEMBL23770415 0.83 ADORA2A (0.34) ADORA2AADORA1SMN1; SMN2GAADPP4
SCHEMBL23770545 0.82 DHFR (0.30)
SCHEMBL23770772 0.82 CSNK2A2 (0.33)
SCHEMBL23770680 0.80 CTSA (0.31)
SCHEMBL23770756 0.80 BACE1 (0.36) ALDH1A1DPP4
SCHEMBL23770602 0.79 NOS3 (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3504194-B1 N-(PYRIDIN-2-YL)PYRIDINE-SULFONAMIDE DERIVATIVES AND THEIR USE IN THE TREATMENT OF DISEASE NOVARTIS AG (CH) 2021-08-18 EP disclosed