SCHEMBL23792833

SCHEMBL23792833

C=C(CC(C)(C)C)c1ccc(N)cc1

nearest known ligand 0.41

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 4/20 0.39
LMNA P02545 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
MAOA P21397 1/20 0.37
MASP2 O00187 1/20 0.37
PLAU P00749 1/20 0.37
THPO P40225 1/20 0.37
EPHX2 P34913 1/20 0.37
F2 P00734 1/20 0.35
PRSS1 P07477 1/20 0.35
APEX1 P27695 1/20 0.35
PRSS3 P35030 1/20 0.35
ESR1 P03372 2/20 0.35
ESR2 Q92731 2/20 0.35
ESRRG P62508 1/20 0.35
THRA P10827 1/20 0.34
THRB P10828 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3144723 0.84 NPC1 (0.44) CYP19A1LMNACYP1A2CYP3A4MAOA
SCHEMBL2399414 0.78 MAOA (0.47) MAOA
SCHEMBL11698205 0.76 CYP19A1 (0.54) CYP19A1LMNACYP1A2CYP3A4MAOA
SCHEMBL14041429 0.75 LMNA (0.46) CYP19A1LMNACYP1A2CYP3A4MAOA
SCHEMBL508101 0.75 GSK3B (0.42) CYP19A1LMNAEPHX2
SCHEMBL15868678 0.75 MAOA (0.34) CYP19A1MAOAMASP2PLAUTHPO
SCHEMBL23792863 0.74 HDAC1 (0.47) MAOA
SCHEMBL23793503 0.73 ALDH1A1 (0.37) THRB
SCHEMBL14330440 0.72 CYP19A1 (0.45) CYP19A1LMNACYP1A2CYP3A4MAOA
SCHEMBL10856840 0.71 PHLPP2 (0.43) CYP19A1CYP3A4MAOA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021178907-A1 STAT INHIBITORY COMPOUNDS AND COMPOSITIONS JANPIX, LTD. (US) 2021-09-10 WO disclosed