SCHEMBL2390071

SCHEMBL2390071

CC(=O)Oc1cccc(C=O)c1C

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 2/20 0.56
TLR2 O60603 1/20 0.56
TLR1 Q15399 1/20 0.56
TLR6 Q9Y2C9 1/20 0.56
ACHE P22303 1/20 0.56
ALDH1A1 P00352 3/20 0.45
LMNA P02545 2/20 0.45
PTGDR2 Q9Y5Y4 1/20 0.45
MAPK1 P28482 1/20 0.45
CYP1A2 P05177 1/20 0.45
CYP2C9 P11712 1/20 0.45
CYP2C19 P33261 1/20 0.45
KDM4E B2RXH2 3/20 0.44
HPGD P15428 2/20 0.44
HSD17B10 Q99714 2/20 0.44
ESR1 P03372 1/20 0.44
ITGB3 P05106 1/20 0.44
ITGA2B P08514 1/20 0.44
HMGB1 P09429 1/20 0.44
TSHR P16473 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30331767 1.00 ERN1 (0.56) ERN1TLR2TLR1TLR6ACHE
SCHEMBL870959 0.85 ALDH1A1 (0.55) ERN1TLR2TLR1TLR6ALDH1A1
SCHEMBL11534206 0.84 ERN1 (0.50) ERN1TLR2TLR1TLR6ACHE
SCHEMBL3248320 0.84 ACHE (0.54) ERN1TLR2TLR1TLR6ACHE
SCHEMBL12587484 0.84 ACHE (0.45) ACHEALDH1A1LMNAMAPK1KDM4E
SCHEMBL3864807 0.84 ERN1 (0.68) ERN1TLR2TLR1TLR6ACHE
Benzene SCHEMBL3155472 0.83 ALDH1A1 (0.58) ERN1TLR2TLR1TLR6ALDH1A1
SCHEMBL1959471 0.83 ERN1 (0.53) ERN1TLR2TLR1TLR6ACHE
SCHEMBL544041 0.82 ACHE (0.69) ACHEALDH1A1LMNAMAPK1CYP1A2
SCHEMBL5241671 0.82 MAPK1 (0.57) ERN1TLR2TLR1TLR6ACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105307638-A Photosensitive particles and application thereof in photodynamic therapy and development XUE FUSHENG 2016-02-03 CN disclosed
US-8012964-B2 9-substituted 8-oxoadenine compound DAINIPPON SUMITOMO PHARMA CO., LTD. (JP) 2011-09-06 US disclosed
CN-100439331-C Intermediate of anti-AIDS medicine 'Nelfinavir' and its syntesizing process and application SHANGHAI INST ORGANIC CHEM (CN) 2008-12-03 CN disclosed
US-7217794-B2 Compounds and methods for treatment of thrombosis DAIAMED, INC. (US) 2007-05-15 US disclosed
US-20050215801-A1 Process for preparation of optically active 1-substituted amino-2,3-epoxypropanes, intermediates for synthesis thereof and process for preparation of the intermediates KANEKA CORPORATION (JP) 2005-09-29 US disclosed
EP-1553093-A1 PROCESS FOR PREPARATION OF OPTICALLY ACTIVE 1-SUBSTITUTED AMINO-2,3-EPOXYPROPANES, INTERMEDIATES FOR THE SYNTHESIS THEREOF AND PROCESS FOR PREPARATION OF THE INTERMEDIATES KANEKA CORPORATION (JP) 2005-07-13 EP disclosed
US-20050143317-A1 Compounds and methods for treatment of thrombosis EXITHERA PHARMACEUTICALS LLC 2005-06-30 US disclosed
WO-2004103270-A2 COMPOUNDS AND METHODS FOR TREATMENT OF THROMBOSIS SUNTORY PHARMACEUTICAL RESEARCH LABORATORIES LLC (US) 2004-12-02 WO disclosed
WO-2004089297-A2 COMPOUNDS AND METHODS FOR TREATMENT OF THROMBOSIS SUNTORY PHARMACEUTICAL RESEARCH LABORATORIES, LLC (US) 2004-10-21 WO disclosed
US-6605721-B2 Intermediates for making HIV-protease inhibitors and methods for making HIV-protease inhibitors AGOURON PHARMACEUTICALS, INC. 2003-08-12 US disclosed
US-6512135-B2 2-methyl-3-(protected hydroxy) benzyl chloride; use making nelfinavir mesylate AGOURON PHARMACEUTICALS, INC. 2003-01-28 US disclosed
US-6407285-B1 AS CHEMICAL INTERMEDIATE TO PREPARE NELFINAVIR COMPOUNDS AGOURON PHARMACEUTICALS, INC. 2002-06-18 US disclosed
US-6303786-B1 SALT FORMATION IN A SOLVENT AGOURON PHARMACEUTICALS, INC. 2001-10-16 US disclosed
EP-0927165-A2 INTERMEDIATES FOR MAKING HIV-PROTEASE INHIBITORS AND METHODS OF MAKING HIV-PROTEASE INHIBITORS AGOURON PHARMACEUTICALS, INC. (US) 1999-07-07 EP disclosed
WO-1998009951-A2 INTERMEDIATES FOR MAKING HIV-PROTEASE INHIBITORS AND METHODS OF MAKING HIV-PROTEASE INHIBITORS AGOURON PHARMACEUTICALS, INC. (US) 1998-03-12 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050143317-A1 Compounds and methods for treatment of thrombosis SERPINC1, F11, F13B ERN1 2398/4885TLR2 3685/4885TLR1 4153/4885
US-20050215801-A1 Process for preparation of optically active 1-substituted amino-2,3-epoxypropanes, intermediates for synthesis thereof and process for preparation of the intermediates OXER1, RCC2, CBR3 ERN1 1143/4885TLR2 2792/4885TLR1 1231/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.