SCHEMBL2391787

SCHEMBL2391787

O=CCSc1ccccn1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 4/20 0.61
NPC1 O15118 3/20 0.61
TDP1 Q9NUW8 2/20 0.61
L3MBTL1 Q9Y468 1/20 0.61
ALDH1A1 P00352 5/20 0.51
EHMT2 Q96KQ7 1/20 0.50
EHMT1 Q9H9B1 1/20 0.50
APOBEC3G Q9HC16 1/20 0.50
KMT2A Q03164 2/20 0.47
MAPT P10636 2/20 0.47
MEN1 O00255 1/20 0.47
PKM P14618 1/20 0.47
POLB P06746 2/20 0.46
LMNA P02545 1/20 0.46
HPGD P15428 3/20 0.45
HSD17B10 Q99714 2/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
KDM4E B2RXH2 1/20 0.45
ALOX15 P16050 1/20 0.45
NPSR1 Q6W5P4 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2304577 0.85 NPC1 (0.72) RAB9ANPC1TDP1L3MBTL1ALDH1A1
SCHEMBL2304581 0.85 NPC1 (0.72) RAB9ANPC1TDP1L3MBTL1ALDH1A1
SCHEMBL5580510 0.81 ALDH1A1 (0.57) RAB9ANPC1TDP1L3MBTL1ALDH1A1
SCHEMBL2874801 0.80 NPC1 (0.61) RAB9ANPC1TDP1L3MBTL1ALDH1A1
SCHEMBL3647399 0.80 NPC1 (0.61) RAB9ANPC1TDP1L3MBTL1ALDH1A1
Hydrogen Sulfide SCHEMBL27801563 0.78 NPC1 (0.59) RAB9ANPC1TDP1L3MBTL1ALDH1A1
SCHEMBL12709500 0.77
SCHEMBL4687320 0.77
SCHEMBL7205329 0.76 EHMT2 (0.61) RAB9ANPC1TDP1L3MBTL1ALDH1A1
SCHEMBL28462526 0.76 L3MBTL1 (1.00) RAB9ANPC1TDP1L3MBTL1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-110514752-B Extraction method of additive in paper food packaging material and non-targeted screening method thereof 云南中烟工业有限责任公司 2022-03-11 CN claimed
US-20220340893-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2022-10-27 US disclosed
EP-3000807-B1 MERCAPTONICOTINIC ACID COMPOUND AND PREPARATION METHOD AND USE THEREOF ACAD OF MILITARY MEDICAL SCIENCES (CN) 2021-04-21 EP disclosed
CN-105218632-A As peptide or plan peptide, the Preparation Method And The Use of transglutaminase inhibitor ZEDIRA GMBH 2016-01-06 CN disclosed
US-8471063-B2 Michael systems as transglutaminase inhibitors ZEDIRA GMBH (DE) 2013-06-25 US disclosed
US-20110229568-A1 MICHAEL SYSTEMS AS TRANSGLUTAMINASE INHIBITORS ZEDIRA GMBH (DE) 2011-09-22 US disclosed
US-20100248365-A1 GANGLIOSIDE BIOSYNTHESIS MODULATORS ZACHARON PHARMACEUTICALS, INC. (US) 2010-09-30 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100248365-A1 GANGLIOSIDE BIOSYNTHESIS MODULATORS UGCG, MAGT1, STT3B RAB9A 1124/4885NPC1 622/4885TDP1 3386/4885
US-20110229568-A1 MICHAEL SYSTEMS AS TRANSGLUTAMINASE INHIBITORS TGM2, TGM3, TGM1 RAB9A 1772/4885NPC1 3980/4885TDP1 2440/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.