SCHEMBL23928823

SCHEMBL23928823

CC(C)(C)OC(=O)NC1(O)C=CC(c2ccccc2)=CC1N

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NFKB1 P19838 1/20 0.37
NFKB2 Q00653 1/20 0.37
RELA Q04206 1/20 0.37
CKS1B P61024 3/20 0.34
SKP1 P63208 3/20 0.34
SKP2 Q13309 3/20 0.34
IDO1 P14902 1/20 0.34
ACACB O00763 1/20 0.34
ACACA Q13085 1/20 0.34
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
MEN1 O00255 1/20 0.33
NPC1 O15118 1/20 0.33
GAA P10253 1/20 0.33
RAB9A P51151 1/20 0.33
KMT2A Q03164 1/20 0.33
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA7 P43166 1/20 0.33
CA14 Q9ULX7 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23748573 0.82 SMYD3 (0.32) LMNA
SCHEMBL5983441 0.73 NFKB1 (0.36) NFKB1NFKB2RELACKS1BSKP1
Methane SCHEMBL27537449 0.72 NFKB1 (0.36) NFKB1NFKB2RELACKS1BSKP1
SCHEMBL6852873 0.69 THRB (0.33) LMNA
SCHEMBL28874371 0.69 HTT (0.34) MEN1GAAKMT2AKDM1AMAOB
SCHEMBL28652511 0.69 HTT (0.35) ALDH1A1LMNAMEN1GAAKMT2A
SCHEMBL28716007 0.68 MMP3 (0.31) MAOB
SCHEMBL27485455 0.68 LMNA (0.31) LMNA
SCHEMBL28538107 0.68 LMNA (0.34) LMNA
SCHEMBL28579116 0.68 LMNA (0.34) LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20210332036-A1 PYRIMIDINE AND PYRAZINE HDAC1,2 INHIBITORS REGENACY PHARMACEUTICALS LLC (US) 2021-10-28 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210332036-A1 PYRIMIDINE AND PYRAZINE HDAC1,2 INHIBITORS HDAC1, HDAC2, HDAC11 NFKB1 1793/4885NFKB2 2104/4885RELA 1628/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.