SCHEMBL23971222

SCHEMBL23971222

COC(=O)c1ccc(OC)nc1Br

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 2/20 0.50
POLB P06746 1/20 0.50
TDP1 Q9NUW8 1/20 0.50
NNMT P40261 1/20 0.49
ALDH1A1 P00352 4/20 0.46
KDM4E B2RXH2 3/20 0.46
RAB9A P51151 4/20 0.41
NPC1 O15118 3/20 0.41
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA7 P43166 1/20 0.41
PDK2 Q15119 1/20 0.41
PDK4 Q16654 1/20 0.41
CA9 Q16790 1/20 0.41
CA14 Q9ULX7 1/20 0.41
SMN1; SMN2 Q16637 5/20 0.40
KMT2A Q03164 2/20 0.40
TSHR P16473 3/20 0.40
HPGD P15428 3/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22658874 0.85 L3MBTL1 (0.45) L3MBTL1POLBALDH1A1KDM4ERAB9A
SCHEMBL29587479 0.85 L3MBTL1 (0.45) L3MBTL1POLBALDH1A1KDM4ERAB9A
SCHEMBL28045757 0.84 TDP1 (0.66) L3MBTL1POLBTDP1NNMTALDH1A1
SCHEMBL7902874 0.80 POLB (0.51) L3MBTL1POLBTDP1NNMTALDH1A1
SCHEMBL2473278 0.80 NPC1 (0.43) L3MBTL1ALDH1A1KDM4ERAB9ANPC1
SCHEMBL21041119 0.80 NNMT (0.69) L3MBTL1POLBTDP1NNMTALDH1A1
SCHEMBL11605385 0.80 TDP1 (0.71) L3MBTL1POLBTDP1NNMTALDH1A1
SCHEMBL30527055 0.79 POLB (0.47) L3MBTL1POLBTDP1NNMTALDH1A1
SCHEMBL21041142 0.79 POLB (0.47) L3MBTL1POLBTDP1NNMTALDH1A1
SCHEMBL23970964 0.79 TUBB4A (0.51) L3MBTL1ALDH1A1KDM4ERAB9ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021222353-A1 MACROCYCLIC INHIBITORS OF PEPTIDYLARGININE DEIMINASES GILEAD SCIENCES, INC. (US) 2021-11-04 WO disclosed