SCHEMBL2404367

SCHEMBL2404367

C[N][C@H](C)c1ccccc1F

nearest known ligand 0.44

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HSD11B1 P28845 8/20 0.44
CYP3A4 P08684 2/20 0.38
IDO1 P14902 1/20 0.37
TDO2 P48775 1/20 0.37
CES2 O00748 1/20 0.37
CES1 P23141 1/20 0.37
ACHE P22303 1/20 0.37
MEN1 O00255 1/20 0.37
ALDH1A1 P00352 1/20 0.37
MAPT P10636 1/20 0.37
CYP2C9 P11712 1/20 0.37
KMT2A Q03164 1/20 0.37
MAPKAPK2 P49137 1/20 0.34
GABRA1 P14867 1/20 0.33
GABRB2 P47870 1/20 0.33
GAA P10253 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20621908 0.76 ACHE (0.40) HSD11B1CYP3A4IDO1TDO2CES2
SCHEMBL31852251 0.75 GABRA1 (0.50) CYP3A4IDO1TDO2CES2CES1
SCHEMBL84442 0.75 GABRA1 (0.50) CYP3A4IDO1TDO2CES2CES1
SCHEMBL15903486 0.75 ACHE (0.43) HSD11B1CYP3A4IDO1TDO2CES2
SCHEMBL2401904 0.74 CES2 (0.36) CES2CES1ACHEALDH1A1GAA
SCHEMBL2402247 0.74 ESR1 (0.48) CYP3A4ACHEALDH1A1CYP2C9GABRA1
SCHEMBL4199089 0.73 GABRA1 (0.60) CYP3A4MEN1ALDH1A1MAPTCYP2C9
SCHEMBL2400168 0.73 HSD11B1 (0.44) HSD11B1CYP3A4IDO1TDO2ALDH1A1
SCHEMBL2400751 0.73 HSD11B1 (0.44) HSD11B1CYP3A4IDO1TDO2ALDH1A1
SCHEMBL2401009 0.72 HSD11B1 (0.48) HSD11B1IDO1TDO2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8835427-B2 Fungicidal heterocyclic compounds E I DU PONT DE NEMOURS AND COMPANY (US) 2014-09-16 US disclosed
EP-2358709-B1 FUNGICIDAL HETEROCYCLIC COMPOUNDS DU PONT (US) 2014-01-22 EP disclosed
US-8618137-B2 Fungicidal heterocyclic compounds E I DU PONT DE NEMOURS AND COMPANY (US) 2013-12-31 US disclosed
US-20120309752-A1 FUNGICIDAL HETEROCYCLIC COMPOUNDS E I DU PONT DE NEMOURS AND COMPANY (US) 2012-12-06 US disclosed
US-20110224258-A1 FUNGICIDAL HETEROCYCLIC COMPOUNDS E.I. DU PONT DE NEMOURS AND COMPANY (DE) 2011-09-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110224258-A1 FUNGICIDAL HETEROCYCLIC COMPOUNDS NOX1, XDH, CBR1 HSD11B1 426/4885CYP3A4 91/4885IDO1 226/4885
US-20120309752-A1 FUNGICIDAL HETEROCYCLIC COMPOUNDS CYP1B1, NOX3, CYP1A1 HSD11B1 424/4885CYP3A4 68/4885IDO1 183/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.