SCHEMBL24050331

SCHEMBL24050331

C=CC(=C)c1ccccc1N(C)C

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 3/20 0.53
MAPT P10636 3/20 0.53
TSHR P16473 2/20 0.53
ALDH1A1 P00352 2/20 0.53
TP53 P04637 1/20 0.53
SMN1; SMN2 Q16637 1/20 0.53
CNR2 P34972 2/20 0.38
PTPN1 P18031 2/20 0.34
KDM4E B2RXH2 2/20 0.34
CHEK1 O14757 1/20 0.34
NEK2 P51955 1/20 0.34
LIMK1 P53667 1/20 0.34
DYRK1A Q13627 1/20 0.34
CLK4 Q9HAZ1 1/20 0.34
KMT2A Q03164 2/20 0.33
MEN1 O00255 1/20 0.33
EP300 Q09472 1/20 0.33
KAT2B Q92831 1/20 0.33
KAT8 Q9H7Z6 1/20 0.33
BRD4 O60885 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29365484 0.79 MAPT (0.61) GAAMAPTTSHRALDH1A1TP53
SCHEMBL8924902 0.79 MAPT (0.61) GAAMAPTTSHRALDH1A1TP53
SCHEMBL10367206 0.78 MAPT (0.62) GAAMAPTTSHRALDH1A1TP53
SCHEMBL8578207 0.77 GAA (0.59) GAAMAPTTSHRALDH1A1TP53
SCHEMBL24050095 0.76 GAA (0.48) GAAMAPTTSHRALDH1A1TP53
SCHEMBL25724853 0.76 ALDH1A1 (0.33) GAAMAPTTSHRALDH1A1TP53
SCHEMBL2267690 0.75 MAPT (0.57) GAAMAPTTSHRALDH1A1TP53
SCHEMBL19685318 0.73 MAPT (0.55) GAAMAPTTSHRALDH1A1TP53
SCHEMBL2491643 0.73 MAPT (0.67) GAAMAPTTSHRALDH1A1TP53
SCHEMBL5965069 0.72 MAOA (0.44) TSHRALDH1A1TP53SMN1; SMN2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3713927-B1 PYRIDINONE DERIVATIVES AND THEIR USE AS SELECTIVE ALK-2 INHIBITORS NOVARTIS AG (CH) 2021-12-15 EP disclosed
WO-2021236489-A1 BIOMASS DERIVED DIKETONES AS EFFICIENT VISIBLE LIGHT PHOTOINITIATORS BOWLING GREEN STATE UNIVERSITY (US) 2021-11-25 WO disclosed