SCHEMBL2405923

SCHEMBL2405923

COC(=O)C(C(=O)c1ccc(F)cc1)c1ccc(O)c(Br)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FOLH1 Q04609 1/20 0.42
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
NPC1 O15118 2/20 0.39
MAPT P10636 2/20 0.39
HTT P42858 2/20 0.39
RAB9A P51151 2/20 0.39
KDM4E B2RXH2 2/20 0.39
USP2 O75604 1/20 0.39
TP53 P04637 1/20 0.39
ALOX15 P16050 1/20 0.39
ALOX12 P18054 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
HSD17B10 Q99714 1/20 0.39
ESR1 P03372 1/20 0.39
MAPK1 P28482 1/20 0.37
KCNMA1 Q12791 1/20 0.36
CCR6 P51684 1/20 0.36
HKDC1 Q2TB90 1/20 0.36
GAA P10253 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2402264 0.80 MAPT (0.39) MEN1KMT2ANPC1MAPTHTT
SCHEMBL6479736 0.74 LTA4H (0.47) MEN1KMT2AKDM4EALDH1A1
SCHEMBL6623432 0.74 EPHX2 (0.52)
SCHEMBL31614294 0.73 MT-CO2 (0.55) FOLH1MEN1KMT2AESR1GAA
SCHEMBL8459765 0.73 FOLH1 (0.50) FOLH1MEN1KMT2AALOX15ESR1
SCHEMBL27640937 0.73 MT-CO2 (0.55) FOLH1MEN1KMT2AESR1GAA
SCHEMBL27965732 0.71 FOLH1 (0.49) FOLH1MEN1KMT2AHDAC3HDAC4
SCHEMBL7069500 0.70 FOLH1 (0.50) FOLH1MEN1KMT2AALOX15ESR1
SCHEMBL974872 0.70 RAB9A (0.44) MEN1KMT2ANPC1MAPTHTT
SCHEMBL13228080 0.69 LMNA (0.47) MEN1KMT2AMAPTKDM4ESMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2542545-A1 INHIBITORS OF HEPATITIS C VIRUS NS5B POLYMERASE Merck Sharp & Dohme Corp. (US) 2013-01-09 EP disclosed
WO-2011106992-A1 INHIBITORS OF HEPATITIS C VIRUS NS5B POLYMERASE MERCK SHARP & DOHME CORP. (US) 2011-09-09 WO disclosed