SCHEMBL2408355

SCHEMBL2408355

CN(Cc1cc(-c2cccnc2F)n(S(=O)(=O)c2ccsc2)c1)C(=O)OC(C)(C)C

nearest known ligand 0.33

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
GLS O94925 1/20 0.33
CTSD P07339 5/20 0.33
BACE1 P56817 5/20 0.33
BACE2 Q9Y5Z0 5/20 0.33
HTR2C P28335 4/20 0.33
SLC6A4 P31645 4/20 0.33
KAT6A Q92794 2/20 0.33
KAT5 Q92993 2/20 0.33
MGLL Q99685 1/20 0.31
PDK2 Q15119 1/20 0.31
HTR2A P28223 1/20 0.31
KAT8 Q9H7Z6 2/20 0.31
SQLE Q14534 1/20 0.30
TACR1 P25103 1/20 0.30
SCN8A Q9UQD0 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2415723 0.89 HTR2C (0.39) GLSHTR2CSLC6A4KAT6AKAT5
SCHEMBL2417461 0.89 GLS (0.32) GLSHTR2CSLC6A4SQLE
SCHEMBL2414740 0.88 HTR2C (0.37) HTR2CSLC6A4KAT6AKAT5HTR2A
SCHEMBL5008212 0.88 CTSD (0.34) CTSDBACE1BACE2TACR1
SCHEMBL2409950 0.87 HTR6 (0.38) HTR2CSLC6A4KAT6AKAT5HTR2A
SCHEMBL1278111 0.87 RIPK1 (0.34) HTR2CSLC6A4KAT6AKAT5KAT8
SCHEMBL2412876 0.87 PTGDR2 (0.39) HTR2CSLC6A4KAT6AKAT5PDK2
SCHEMBL1278411 0.86 KAT6A (0.34) GLSHTR2CSLC6A4KAT6AKAT5
SCHEMBL31187457 0.86 KAT8 (0.35) GLSHTR2CSLC6A4KAT6AKAT5
SCHEMBL2411977 0.86 HTR2C (0.33) GLSHTR2CSLC6A4KAT6AKAT5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2364979-A1 Pyrrole compounds Takeda Pharmaceutical Company Limited (JP) 2011-09-14 EP disclosed
EP-2114917-A2 PYRROLE COMPOUNDS Takeda Pharmaceutical Company Limited (JP) 2009-11-11 EP disclosed
WO-2008108380-A2 PYRROLE COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-09-12 WO disclosed