SCHEMBL2412876

SCHEMBL2412876

CN(Cc1cc(-c2cccnc2F)n(S(=O)(=O)c2ccc(F)c(F)c2)c1)C(=O)OC(C)(C)C

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 3/20 0.39
CCKAR P32238 1/20 0.39
ALDH3A1 P30838 1/20 0.36
RORC P51449 4/20 0.35
KAT6A Q92794 2/20 0.35
KAT5 Q92993 2/20 0.35
HTR2C P28335 5/20 0.34
SLC6A4 P31645 5/20 0.34
HTR2A P28223 1/20 0.34
GRM4 Q14833 1/20 0.34
GAA P10253 1/20 0.34
KAT8 Q9H7Z6 1/20 0.32
PDK2 Q15119 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2412420 0.93 GRM4 (0.38) PTGDR2CCKARKAT6AKAT5HTR2C
SCHEMBL2414740 0.91 HTR2C (0.37) RORCKAT6AKAT5HTR2CSLC6A4
SCHEMBL2409950 0.91 HTR6 (0.38) KAT6AKAT5HTR2CSLC6A4HTR2A
SCHEMBL2415723 0.91 HTR2C (0.39) PTGDR2KAT6AKAT5HTR2CSLC6A4
SCHEMBL31187457 0.89 KAT8 (0.35) KAT6AKAT5HTR2CSLC6A4HTR2A
SCHEMBL1278411 0.89 KAT6A (0.34) KAT6AKAT5HTR2CSLC6A4HTR2A
SCHEMBL2409374 0.89 HTR2C (0.40) KAT6AKAT5HTR2CSLC6A4HTR2A
SCHEMBL1278111 0.88 RIPK1 (0.34) PTGDR2KAT6AKAT5HTR2CSLC6A4
SCHEMBL2409152 0.88 ALDH1A1 (0.37) KAT6AKAT5HTR2CSLC6A4GAA
SCHEMBL31187449 0.88 MET (0.42) HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2364979-A1 Pyrrole compounds Takeda Pharmaceutical Company Limited (JP) 2011-09-14 EP disclosed
EP-2114917-A2 PYRROLE COMPOUNDS Takeda Pharmaceutical Company Limited (JP) 2009-11-11 EP disclosed
WO-2008108380-A2 PYRROLE COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-09-12 WO disclosed