SCHEMBL2412428

SCHEMBL2412428

CC(C)(C)C(Cc1cn(S(=O)(=O)c2cccc(F)c2)c(-c2cccnc2Cl)c1F)NC(=O)O

nearest known ligand 0.35

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
NFE2L2 Q16236 3/20 0.35
HTR6 P50406 11/20 0.34
PTGDR2 Q9Y5Y4 3/20 0.34
IDE P14735 1/20 0.32
HTR2A P28223 1/20 0.32
HTR2C P28335 1/20 0.32
HTR7 P34969 1/20 0.32
DHODH Q02127 1/20 0.32
PTGDR Q13258 1/20 0.32
CYP3A4 P08684 1/20 0.32
SCN9A Q15858 1/20 0.32
SCN10A Q9Y5Y9 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2412415 0.93 PTGDR2 (0.34) HTR6PTGDR2HTR2AHTR7DHODH
SCHEMBL2412127 0.91 MET (0.39) NFE2L2HTR6PTGDR2HTR2A
SCHEMBL2408070 0.90 PPME1 (0.34) HTR6PTGDR2
SCHEMBL2408861 0.90 FPR1 (0.33) IDE
SCHEMBL2409871 0.88 PTGDR2 (0.33) HTR6PTGDR2IDEHTR2AHTR2C
SCHEMBL2409033 0.85 PTGDR2 (0.32) PTGDR2
SCHEMBL2407582 0.85 MET (0.38) PTGDR2
SCHEMBL2412156 0.84 DCTPP1 (0.32) PTGDR2
SCHEMBL2415885 0.83 ADAMTS4 (0.31) PTGDR2DHODH
SCHEMBL2412351 0.83 MET (0.40) NFE2L2HTR6PTGDR2HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2364979-A1 Pyrrole compounds Takeda Pharmaceutical Company Limited (JP) 2011-09-14 EP disclosed