SCHEMBL24136206

SCHEMBL24136206

COc1ccc(F)c2cc(C)n(I)c12

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 3/20 0.35
NQO2 P16083 3/20 0.35
TUBB1 Q9H4B7 3/20 0.34
LMNA P02545 2/20 0.33
KDM4E B2RXH2 2/20 0.33
ALDH1A1 P00352 2/20 0.33
ACHE P22303 1/20 0.33
NFE2L2 Q16236 1/20 0.33
MAPK1 P28482 1/20 0.33
HTT P42858 1/20 0.33
RAB9A P51151 1/20 0.33
TSHR P16473 1/20 0.33
MAPT P10636 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
NR4A1 P22736 1/20 0.33
THRB P10828 1/20 0.32
HPGD P15428 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
TRPA1 O75762 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL24136189 0.87 MEN1 (0.35) CYP19A1NQO2TUBB1LMNAKDM4E
SCHEMBL22434778 0.81 CYP19A1 (0.44) CYP19A1NQO2TUBB1LMNAKDM4E
SCHEMBL20504816 0.75 HASPIN (0.42) CYP19A1NQO2KDM4EMAPK1MAPT
SCHEMBL24136153 0.73 PDE2A (0.35)
SCHEMBL24136193 0.72 HRH4 (0.33) CYP1A2
SCHEMBL22434669 0.71 CYP19A1 (0.40) CYP19A1NQO2TUBB1LMNAKDM4E
SCHEMBL24136162 0.70 CYP11B1 (0.35)
SCHEMBL24136161 0.69
SCHEMBL24136199 0.69 HTR2A (0.43) CYP19A1NQO2LMNAKDM4EALDH1A1
SCHEMBL24136151 0.69 ACLY (0.34)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3928836-A1 N-SUBSTITUTED INDOLE DERIVATIVES AS PGE2 RECEPTOR MODULATORS Idorsia Pharmaceuticals Ltd (CH) 2021-12-29 EP disclosed